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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
58 Results for "
SERM
" in MedChemExpress (MCE) Product Catalog:
Products (58)
58 Results for "SERM" in MCE Product Catalog:
Cat. No.: HY-B0005AS
Synonyms: Z-Toremifene-d6; NK 622-d6 free base; FC-1157a-d6 free base
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LY117018, a Raloxifene analog, is a selective estrogen receptor modulator. LY117018 exerts antiproliferative effects on breast cancer cell lines .
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LY117018 TFA, a Raloxifene analog, is a selective estrogen receptor modulator. LY117018 TFA exerts antiproliferative effects on breast cancer cell lines .
Cat. No.: HY-116896R
CAS No.: 63676-25-5
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LY117018 (Standard) is the analytical standard of LY117018. This product is intended for research and analytical applications. LY117018, a Raloxifene analog, is a selective estrogen receptor modulator. LY117018 exerts antiproliferative effects on breast cancer cell lines .
Cat. No.: HY-B0723S2
Synonyms: FC-1271a-d5
Cat. No.: HY-B0005S
CAS No.: 1246833-71-5
Cat. No.: HY-B0005R
CAS No.: 89778-27-8
Synonyms: Z-Toremifene citrate (Standard); NK 622 (Standard); FC-1157a (Standard)
Toremifene (citrate) (Standard) is the analytical standard of Toremifene (citrate). This product is intended for research and analytical applications. Toremifene citrate (Z-Toremifene citrate) is a second-generation selective estrogen-receptor modulator (SERM) in development for the prevention of osteoporosis. Toremifene citrate also potent inhibits infectious EBOV Zaire and Marburg (MARV) with IC50 of 0.07 µM and 2.6 µM, respectively .
Cat. No.: HY-125091
CAS No.: 648904-56-7
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LY2066948 is a selective and orally active estrogen receptor modulator (SERM). LY2066948 has high affinity for estrogen receptors ERα and ERβ (Ki: 0.51 and 1.36 nM respectively) and shows potent antiestrogenic activity. LY2066948 blocks uterine weight gain induced by Ethynyl estradiol (HY-B0216) in immature rats. LY2066948 can be used for research of uterine fibroids and myomas .
Cat. No.: HY-A0031S
CAS No.: 1133695-49-4
Synonyms: TSE-424-d4
Cat. No.: HY-A0031S2
CAS No.: 1795027-71-2
Synonyms: TSE-424-d4 acetate
Cat. No.: HY-13757AS1
CAS No.: 508201-30-7
Synonyms: ICI 47699-d3; (Z)-Tamoxifen-d3; trans-Tamoxifen-d3
Cat. No.: HY-W778408
CAS No.: 1346606-38-9
Synonyms: ICI 47699-13C6; (Z)-Tamoxifen-13C6; trans-Tamoxifen-13C6
Cat. No.: HY-179232
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ERα antagonist 2 (Compound 5b) is an ER-α antagonist with an IC50 value of 1729 nM. ERα antagonist 2 exhibits significant inhibitory activity against breast cancer cell lines, and is still effective against ER-negative cells (MDA-MB-231), suggesting the existence of ER-independent pathways. ERα antagonist 2 can be used for the study of breast cancer .
Cat. No.: HY-Z0833
CAS No.: 1174289-22-5
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Bazedoxifene N-Oxide is the oxidative degradation product of selective estrogen receptor modulator (SERM) Bazedoxifene .
Cat. No.: HY-U00178R
CAS No.: 116057-75-1
Synonyms: CB7432 (Standard)
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Idoxifene (CB7432) is a novel tissue-specific selective estrogen receptor modulator (SERM).
Cat. No.: HY-A0037R
CAS No.: 180916-16-9
Synonyms: CP-336156 (Standard)
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Lasofoxifene (Standard) is the analytical standard of Lasofoxifene. This product is intended for research and analytical applications. Lasofoxifene (CP-336156) is an orally active and selective estrogen receptor modulator (SERM). Lasofoxifene exhibits an anti-osteoporotic function and also inhibits primary tumor growth and metastases. Lasofoxifene can be used for research of breast cancer and postmenopausal osteoporosis .
Cat. No.: HY-N17536
CAS No.: 1124321-96-5
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Cat. No.: HY-13757AS2
CAS No.: 3047060-10-3
Synonyms: ICI 47699-d2; (Z)-Tamoxifen-d2; trans-Tamoxifen-d2
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
