5 Results for "

Adenosine receptor antagonist-7

" in MedChemExpress (MCE) Product Catalog:
Products (5)

5 Results for "Adenosine receptor antagonist-7" in MCE Product Catalog:

Cat. No.: HY-179248
CAS No.: 2570904-69-5
Research Areas:  

Cancer

Adenosine receptor antagonist 7 is an orally active triple A1/A2A/A2B adenosine receptor antagonist with Ki values of 1.5, 0.6 and 21 nM. Adenosine receptor antagonist 7 shows potent inhibitory activity (IC50 = 0.8 nM) of cAMP production in A2AR-HEK293 cells. Adenosine receptor antagonist 7 can enhance infiltration of effector T cells and increase the CD8+/Treg ratio companied with Avelumab (HY-108730). Adenosine receptor antagonist 7can be used for the research of cancer, such as colon cancer .
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Cat. No.: HY-W017163
CAS No.: 552-62-5
7-Methylxanthine is an orally active methyl derivative of xanthine and a non-selective adenosine receptor antagonist. 7-Methylxanthine is also one of the purine components of human urinary calculi. 7-Methylxanthine has anti-myopia activity .
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Cat. No.: HY-174986
CAS No.: 2173508-07-9
Target:  

CGRP Receptor

Research Areas:  

Cardiovascular Disease

CGRP antagonist 7 is a potent calcitonin gene-related peptide receptor (CGRP) antagonist with a Ki of 0.029 nM. CGRP antagonist 7 Inhibit the production of cyclic adenosine monophosphate (cAMP) with an IC50 of 1.5 nM. CGRP antagonist 7 can be used for the study of migraine .
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Cat. No.: HY-182432
CAS No.: 2672534-18-6
Target:  

Adenosine Receptor

Research Areas:  

Cancer

A3AR antagonist-7 is a conjugable human A3 adenosine receptor (A3AR) antagonist with a Ki value of 31.8 nM. A3AR antagonist-7 is applicable to the research of melanoma, breast cancer and colorectal cancer .
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Cat. No.: HY-W017163R
CAS No.: 552-62-5
7-Methylxanthine (Standard) is the analytical standard of 7-Methylxanthine. This product is intended for research and analytical applications. 7-Methylxanthine is an orally active methyl derivative of xanthine and a non-selective adenosine receptor antagonist. 7-Methylxanthine is also one of the purine components of human urinary calculi. 7-Methylxanthine has anti-myopia activity .
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