3 Results for "

Aurora A inhibitor-2

" in MedChemExpress (MCE) Product Catalog:
Products (3)

3 Results for "Aurora A inhibitor-2" in MCE Product Catalog:

Cat. No.: HY-146037
CAS No.: 2412144-74-0
Target:  

Apoptosis Aurora Kinase

Research Areas:  

Cancer

Aurora A inhibitor 2 (Compound 16h) is a potent Aurora A kinase inhibitor with an IC50 of 21.94 nM. Aurora A inhibitor 2 induces caspase-dependent apoptosis in MDA-MB-231 cells .
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1
1 Cited Publications
Cat. No.: HY-156863
CAS No.: 2592436-21-8
Purity:  98.88%
GRK2 Inhibitor 2 is an orally active and selective G protein-coupled receptor kinase 2 (GRK) inhibitor with an IC50 of 19 nM. GRK2 Inhibitor 2 also inhibits Aurora-A with an IC50 of 137 nM. GRK2 Inhibitor 2 can be used in the study of congestive heart failure (HF) .
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Cat. No.: HY-112355
CAS No.: 331770-21-9
Purity:  99.08%
Target:  

Aurora Kinase

Research Areas:  

Cancer

Aurora kinase inhibitor-2 is a selective and ATP-competitive Aurora kinase inhibitor with IC50s of 310 nM and 240 nM for Aurora A and Aurora B, respectively .
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