2592436-21-8
2592436-21-8
Chemical Structure
GRK2 Inhibitor 2
- CAS 番号: 2592436-21-8
- Formula:C19H16N4O2
- Molecular Weight:332.36
InChIKey: CYINSAOYPJZRPS-UHFFFAOYSA-N
SMILES: O=C1C2=C(C=NN1CC3=CC(OC)=CC=C3)C=CC(C4=CNN=C4)=C2
Biological Activity: GRK2 Inhibitor 2 is an orally active and selective G protein-coupled receptor kinase 2 (GRK) inhibitor with an IC50 of 19 nM. GRK2 Inhibitor 2 also inhibits Aurora-A with an IC50 of 137 nM. GRK2 Inhibitor 2 can be used in the study of congestive heart failure (HF)[1].
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GRK2 Inhibitor 2 | 99.92% | GRK2 Inhibitor 2 is an orally active and selective G protein-coupled receptor kinase 2 (GRK) inhibitor with an IC50 of 19 nM. GRK2 Inhibitor 2 also inhibits Aurora-A with an IC50 of 137 nM. GRK2 Inhibitor 2 can be used in the study of congestive heart failure (HF). | ||||||||||||||||||||
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