39 Results for "

Lidocaine

" in MedChemExpress (MCE) Product Catalog:
Products (39)

39 Results for "Lidocaine" in MCE Product Catalog:

23
23 Publications Verification
Cat. No.: HY-B0185
CAS No.: 137-58-6
Synonyms: Lignocaine
Lidocaine (Lignocaine) inhibits sodium channels involving complex voltage and using dependence . Lidocaine decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine is an amide derivative and has potential for the research of ventricular arrhythmia .
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23
23 Publications Verification
Cat. No.: HY-B0185A
CAS No.: 73-78-9
Synonyms: Lignocaine hydrochloride
Lidocaine hydrochloride (Lignocaine hydrochloride) inhibits sodium channels involving complex voltage and using dependence . Lidocaine hydrochloride decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine hydrochloride is an amide derivative and a agent to treat ventricular arrhythmia and an effective tumor-inhibitor .
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23
23 Publications Verification
Cat. No.: HY-B0185B
CAS No.: 6108-05-0
Synonyms: Lignocaine hydrochloride hydrate
Lidocaine (Lignocaine) hydrochloride hydrate inhibits sodium channels involving complex voltage and using dependence. Lidocaine hydrochloride hydrate decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine hydrochloride hydrate is an amide derivative and has potential for the research of ventricular arrhythmia .
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3
3 Cited Publications
Cat. No.: HY-66012
CAS No.: 5875-06-9
Synonyms: Proxymetacaine hydrochloride
Target:  

Sodium Channel

Research Areas:  

Neurological Disease

Proparacaine (Proxymetacaine) hydrochloride is a local anesthetic. Proparacaine hydrochloride blocks voltage-gated sodium channels on neuronal cell membranes, thereby inhibiting signal conduction and nociceptive signal transmission. Proparacaine hydrochloride blocks nociceptive signals in the eye and induces ocular muscle relaxation to reduce eye movement during surgery. Proparacaine hydrochloride is used in research related to cataracts .
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Cat. No.: HY-B0185S1
CAS No.: 851528-09-1
Lidocaine-d10 is the deuterium labeled Lidocaine. Lidocaine (Lignocaine) inhibits sodium channels involving complex voltage and using dependence . Lidocaine decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine is an amide derivative and has potential for the research of ventricular arrhythmia .
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Cat. No.: HY-124098
CAS No.: 2903-45-9
Purity:  99.92%
Synonyms: Lidocaine N-oxide
Research Areas:  

Cardiovascular Disease

Lignocaine N-oxide (Lidocaine N-oxide) is a hypoxia-activated prodrug of lidocaine (HY-B0185). Lignocaine N-oxide exerts exactly the same sodium current-blocking effect as lidocaine only when it is converted to lidocaine under ischemic conditions. Lignocaine N-oxide possesses antiarrhythmic activity against ischemia-induced ventricular fibrillation. Lignocaine N-oxide can be used in studies related to ischemia-induced ventricular fibrillation .
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Cat. No.: HY-B0185AS
CAS No.: 1189959-13-4
Lidocaine-d10 (hydrochloride) is the deuterium labeled Lidocaine hydrochloride. Lidocaine hydrochloride (Lignocaine hydrochloride) inhibits sodium channels involving complex voltage and using dependence . Lidocaine hydrochloride decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine hydrochloride, an amide derivative, has the potential for the research of the ventricular arrhythmia .
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Cat. No.: HY-B0185R
CAS No.: 137-58-6
Synonyms: Lignocaine (Standard)
Lidocaine (Standard) is the analytical standard of Lidocaine. This product is intended for research and analytical applications. Lidocaine (Lignocaine) inhibits sodium channels involving complex voltage and using dependence . Lidocaine decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine is an amide derivative and has potential for the research of ventricular arrhythmia .
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Cat. No.: HY-W357818
CAS No.: 18865-38-8
Synonyms: GX
Glycinexylidide (GX) is the active metabolite of Lidocaine. Lidocaine is a local agent that can suppress or relieve pain, that inhibits sodium channels involving complex voltage and dependence. Lidocaine also reduces the growth, migration and invasion of gastric cancer cells. Glycinexylidide has research potential for use in anesthesia, cancer, and cardiovascular disease .
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Cat. No.: HY-114914
CAS No.: 34604-55-2
Target:  

Endogenous Metabolite

Research Areas:  

Cardiovascular Disease

3-Hydroxylidocaine is the major metabolite of Lidocaine (HY-B0185) in rats and sheep .
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Cat. No.: HY-106372A
CAS No.: 1042-42-8
Purity:  99.74%
Synonyms: QX 572; RSD 931
Carcainium chloride (QX 572) is a quaternary derivative of Lidocaine. Antitussive effect .
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Cat. No.: HY-B0185AS1
CAS No.: 2517378-96-8
Synonyms: Lignocaine-d6 hydrochloride
Lidocaine-d6 (hydrochloride) is deuterium labeled Lidocaine (hydrochloride). Lidocaine hydrochloride (Lignocaine hydrochloride) inhibits sodium channels involving complex voltage and using dependence . Lidocaine hydrochloride decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine hydrochloride is an amide derivative and a agent to treat ventricular arrhythmia and an effective tumor-inhibitor .
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Cat. No.: HY-118167
CAS No.: 7728-40-7
Synonyms: MEGX; NorLidocaine
Target:  

Drug Metabolite

Research Areas:  

Metabolic Disease

Monoethylglycinexylidide (MEGX; Norlidocaine) is the major metabolite of Lidocaine (HY-B0185), produced via oxidative metabolism by cytochrome P-450 enzymes in the liver. Monoethylglycinexylidide can be used for research on liver cirrhosis .
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Cat. No.: HY-W099331
CAS No.: 7729-94-4
Synonyms: MEGX hydrochloride; NorLidocaine hydrochloride
Target:  

Drug Metabolite

Research Areas:  

Metabolic Disease

Monoethylglycinexylidide hydrochloride (MEGX hydrochloride; Norlidocaine hydrochloride) is the major metabolite of Lidocaine (HY-B0185), produced via oxidative metabolism by cytochrome P-450 enzymes in the liver. Monoethylglycinexylidide hydrochloride can be used for research on liver cirrhosis .
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Cat. No.: HY-B0185S
CAS No.: 851528-10-4
N-Oxide Lidocaine-d10 is the deuterium labeled Lidocaine. Lidocaine (Lignocaine) inhibits sodium channels involving complex voltage and using dependence . Lidocaine decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine is an amide derivative and has potential for the research of ventricular arrhythmia .
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Cat. No.: HY-Z6535
CAS No.: 857170-72-0
Target:  

Drug Intermediate

Research Areas:  

Others

Lidocaine impurity 12 is an impurity of Lidocaine (HY-B0185).
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Cat. No.: HY-B0185G
CAS No.: 137-58-6
Synonyms: Lignocaine (GMP)
Lidocaine (GMP) is Lidocaine (HY-B0185) produced by using GMP guidelines. GMP small molecules work appropriately as an auxiliary reagent for cell therapy manufacture. Lidocaine inhibits sodium channels involving complex voltage and using dependence . Lidocaine decreases growth, migration and invasion of gastric carcinoma cells via up-regulating miR-145 expression and further inactivation of MEK/ERK and NF-κB signaling pathways. Lidocaine is an amide derivative and has potential for the research of ventricular arrhythmia .
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Cat. No.: HY-B1798
CAS No.: 41708-72-9
Target:  

Sodium Channel

Research Areas:  

Cardiovascular Disease

Tocainide hydrochloride is an orally activesodium channel blocker, it blocks the sodium channels in the pain-producing foci in the nerve membranes. Tocainide hydrochloride is a primary amine analog of lidocaine, can be used for the treatment of tinnitus .
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Cat. No.: HY-101361
CAS No.: 1462-71-1
Synonyms: MethylLidocaine iodide
Target:  

Drug Derivative

Research Areas:  

Neurological Disease

Lidocaine methiodide (Methyllidocaine iodide) is a potent antiarrythmic agent, and is a derivative of Lidocaine (HY-B0185). Lidocaine methiodide can be used for the research of ventricular arrhythmias produced by coronary occlusion .
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Cat. No.: HY-145482
CAS No.: 21236-54-4
Purity:  96.07%
Target:  

Drug Metabolite

Research Areas:  

Neurological Disease

W3601 is the impurity of Lidocaine. W3601 exhibits nerve blocking activity with the pKa of 7.4 .
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