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10 Results for "
Reboxetine mesylate
" in MedChemExpress (MCE) Product Catalog:
Products (10)
10 Results for "Reboxetine mesylate" in MCE Product Catalog:
2
2 Cited Publications
Synonyms: FCE20124 mesylate; PNU155950E mesylate
Target:
Forschungsgebiete:
Reboxetine mesylate (FCE20124 mesylate) is a potent, selective, and specific noradrenaline reuptake inhibitor (NARI) for the research of depression. Reboxetine mesylate inhibits the uptake of norepinephrine, with a Ki of 8 nM .
Art. -Nr.: HY-14790
CAS. Nr.: 98819-76-2
Synonyms: (S,S)-(+)-Reboxetine
Target:
Esreboxetine ((S,S)-Reboxetine) is a selective norepinephrine transporter (NET) inhibitor, with a pIC50 of 9.6 and a pKi of 9.2 in rats, and it can cross the blood-brain barrier. Esreboxetine increases urethral closure pressure and urethral resistance in rats. Esreboxetine is applicable to research related to inflammatory pain and stress urinary incontinence .
Art. -Nr.: HY-14560
CAS. Nr.: 71620-89-8
Target:
Forschungsgebiete:
Reboxetine is an orally active, potent and selective noradrenaline uptake blocker. Reboxetine can be used for antidepressant research .
Art. -Nr.: HY-14560A
CAS. Nr.: 105017-39-8
Synonyms: (R,R)-FCE20124 mesylate; (R,R)-PNU155950E mesylate; (R,R)-(-)-Reboxetine mesylate
Target:
Forschungsgebiete:
(R,R)-Reboxetine mesylate is an antidepressant agent with great bioavailability. (R,R)-Reboxetine is the enantiomer of Reboxetine, which is a selective noradrenaline reuptake inhibitor. Reboxetine consists of (R,R) and (S,S) enantiomer, has low affinity for alpha-adrenergic and muscarinic receptors and low toxicity in animals .
Art. -Nr.: HY-14560CR
CAS. Nr.: 98769-84-7
Synonyms: FCE20124 mesylate (Standard); PNU155950E mesylate (Standard)
Forschungsgebiete:
Reboxetine (mesylate) (Standard) is the analytical standard of Reboxetine (mesylate). This product is intended for research and analytical applications. Reboxetine mesylate (FCE20124 mesylate) is a potent, selective, and specific noradrenaline reuptake inhibitor (NARI) for the research of depression. Reboxetine mesylate inhibits the uptake of norepinephrine, with a Ki of 8 nM .
Art. -Nr.: HY-186094
CAS. Nr.: 105018-14-2
Target:
Forschungsgebiete:
(S,S)-Demethyl-reboxetine is a key phenolic precursor for the preparation of the PET tracer (S,S)-[ 11C]-MeNER. (S,S)-Demethyl-reboxetine is also the demethylated derivative of Reboxetine (HY-14560). Efficient synthesis of the norepinephrine transporter (NET)-targeted tracer is achieved through 11C methylation of (S,S)-Demethyl-reboxetine. (S,S)-Demethyl-reboxetine serves as a core raw material for the synthesis of radiopharmaceuticals related to NET imaging .
Art. -Nr.: HY-186093
CAS. Nr.: 252570-31-3
Target:
Forschungsgebiete:
(S,S)-Reboxetine-OH is a phenol compound. (S,S)-Reboxetine-OH can be used to synthesize norepinephrine transporter ligand .
Art. -Nr.: HY-14790A
CAS. Nr.: 635724-55-9
Synonyms: PNU-165442G; (S,S)-Reboxetine succinate
Target:
Forschungsgebiete:
Esreboxetine succinate (PNU-165442G; (S,S)-Reboxetine succinate) is a selective norepinephrine transporter (NET) inhibitor, with a pIC50 of 9.6 and a pKi of 9.2 in rats, and it can cross the blood-brain barrier. Esreboxetine succinate increases urethral closure pressure and urethral resistance in rats. Esreboxetine succinate is applicable to research related to inflammatory pain and stress urinary incontinence .
Art. -Nr.: HY-183453
CAS. Nr.: 351330-75-1
Target:
Forschungsgebiete:
O-Desethylreboxetine is the major metabolite of Reboxetine (HY-14560), which is catalyzed by the CYP3A4 enzyme. O-Desethylreboxetine can be used in depression-related research .
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Protocols
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