Scientific Reviews
Product Guides
Blogs
Topics
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
49 Results for "
Somatostatin receptor agonist
" in MedChemExpress (MCE) Product Catalog:
Products (49)
49 Results for "Somatostatin receptor agonist" in MCE Product Catalog:
17
Target:
Research Areas:
Cardiovascular Disease Inflammation/Immunology Endocrinology Cancer
6
Target:
Research Areas:
6
Target:
Research Areas:
Pasireotide (SOM230) ditrifluoroacetate, a long-acting cyclohexapeptide somatostatin analogue, can improve agonist activity at somatostatin receptors (subtypes sst1/2/3/4/5, pKi=8.2/9.0/9.1/<7.0/9.9, respectively). Pasireotide ditrifluoroacetate exhibits antisecretory, antiproliferative, and proapoptotic activity .
6
Target:
Research Areas:
6
Target:
Research Areas:
2
Target:
Research Areas:
Target:
Research Areas:
Cat. No.: HY-111615
CAS No.: 848647-56-3
Target:
Research Areas:
Synonyms: LY3556050; CNTX-0290
Target:
Research Areas:
Mazisotine (CNTX-0290) is an orally active, non-opioid somatostatin receptor 4 (SSTR4) agonist with an EC50 of 4.7 nM. Mazisotine exerts significant analgesic effects in various nociceptive (inflammatory, osteoarthritic) and neuropathic pain models. Mazisotine can be used for pain research .
Cat. No.: HY-P5362
Research Areas:
Target:
Research Areas:
L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM. L-803087 is >280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice .
Cat. No.: HY-P10137
CAS No.: 1801415-23-5
Synonyms: JR11
Research Areas:
Synonyms: MK-678; L-363586
Target:
Target:
Research Areas:
L-817818 is a potent and subtype-selective agonist of the somatostatin receptor. L-817818 provides a direct approach to defining somatostatin receptor physiological functions
Cat. No.: HY-142699
CAS No.: 1638589-52-2
Target:
Research Areas:
SSTR4 agonist 2 is a potent agonist of somatostatin receptor subtype 4 (SSTR4). SSTR4 pathway inhibits nociceptive and inflammatory processes. SSTR4 agonist 2 has the potential for the research of medical disorders related to SSTR4 (extracted from patent WO2014184275A1, compound 107) .
Target:
Research Areas:
NNC 26-9100 is a selective somatostatin sst4 receptor full agonist (Ki: 6 nM, EC50: 2 nM). NNC 26-9100 decreases total soluble Aβ42, increases brain neprilysin activity and improves learning .
Cat. No.: HY-P0036A
CAS No.: 1607842-55-6
Synonyms: SMS 201-995 dihydrochloride
Target:
Research Areas:
Cat. No.: HY-142701
CAS No.: 2747928-27-2
Target:
Research Areas:
SSTR4 agonist 4 is a somatostatin receptor 4 (SSTR4) agonist. SSTR4 agonist 4 functionally activates SSTR4. SSTR4 agonist 4 has the potential for the research of pain .
Synonyms: MK 678 acetate; L 36358 acetate
Target:
Research Areas:
Cardiovascular Disease Neurological Disease Metabolic Disease
Cat. No.: HY-P1207
CAS No.: 133073-82-2
Target:
Research Areas:
-
-
Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
