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Cat. No.: HY-168250

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trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl

trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl is a E3 ligase ligand-linker conjugate, and can be used for synthesis of PROTACs, such as PROTAC BRM/BRG1 degrader-2 (HY-168247).

For research use only. We do not sell to patients.

Formula: C₃₄H₄₃ClN₆O₄S
Molecular Weight:667.26

Storage:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (270 KB)

trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl Chemical Structure

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Use of MCE Products

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Biological Activity

Description

trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl is a E3 ligase ligand-linker conjugate, and can be used for synthesis of PROTACs, such as PROTAC BRM/BRG1 degrader-2 (HY-168247)^[1].

All E3 Ligase Ligand-Linker Conjugates Isoforms :

Chemical Information

Molecular Weight 667.26
Formula C₃₄H₄₃ClN₆O₄S
SMILES

CC(C)(C)[C@H](NC([C@H](CC1)CC[C@@H]1C2=CN=C(Cl)N=C2)=O)C(N3C[C@H](O)C[C@H]3C(N[C@H](C4=CC=C(C5=C(C)N=CS5)C=C4)C)=O)=O
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

Purity & Documentation

Select Batch:

Purity: 99.98%

Assay: 99.98%

ee.: 99.98%

Data Sheet (270 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Handling Instructions (2659 KB)

References

[1]. Gu Peng, et al. Brm selective degradation agent compound and use thereof. Patent. WO2023093728

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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Keywords

trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl

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trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl

All E3 Ligase Ligand-Linker Conjugates Isoforms

Biological Activity

Description

Chemical Information

Purity & Documentation

References

Calculators

Help & FAQs

trans-(S,R,S)-AHPC-Me-Amide-cyclohexane-pyrimidine-Cl Related Classifications

HY-168250 Related Classifications

Bioz

Keywords

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