1. Metabolic Enzyme/Protease
  2. Glutaminase
  3. Glutaminase C-IN-1

Glutaminase C-IN-1 (Synonyms: Compound 968)

Cat. No.: HY-12682 Purity: 99.61%
Handling Instructions

Glutaminase C-IN-1 (Compound 968) is an allosteric inhibitor of Glutaminase C that inhibits cancer cell growth without affecting their normal cellular counterparts.

For research use only. We do not sell to patients.

Glutaminase C-IN-1 Chemical Structure

Glutaminase C-IN-1 Chemical Structure

CAS No. : 311795-38-7

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 119 In-stock
Estimated Time of Arrival: December 31
5 mg USD 108 In-stock
Estimated Time of Arrival: December 31
10 mg USD 156 In-stock
Estimated Time of Arrival: December 31
50 mg USD 624 In-stock
Estimated Time of Arrival: December 31
100 mg   Get quote  
200 mg   Get quote  

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Customer Review

Based on 2 publication(s) in Google Scholar

Top Publications Citing Use of Products

Publications Citing Use of MCE Glutaminase C-IN-1

    Glutaminase C-IN-1 purchased from MCE. Usage Cited in: J Hepatol. 2020 May;72(5):909-923.

    Proliferation of HCC-LM3 cells treated with Ctrl, 5 μM 968 alone, 4 μM Sor alone, and combined 5 μM 968 and 4 μM Sor (968+Sor).
    • Biological Activity

    • Purity & Documentation

    • References

    • Customer Review

    Description

    Glutaminase C-IN-1 (Compound 968) is an allosteric inhibitor of Glutaminase C that inhibits cancer cell growth without affecting their normal cellular counterparts.

    Molecular Weight

    475.42

    Formula

    C₂₇H₂₇BrN₂O

    CAS No.

    311795-38-7

    SMILES

    O=C1C(C(C2=CC=C(N(C)C)C(Br)=C2)NC3=C4C5=CC=CC=C5C=C3)=C4CC(C)(C)C1

    Shipping

    Room temperature in continental US; may vary elsewhere.

    Storage
    Powder -20°C 3 years
    4°C 2 years
    In solvent -80°C 6 months
    -20°C 1 month
    Solvent & Solubility
    In Vitro: 

    DMSO : 25 mg/mL (52.59 mM; Need ultrasonic)

    Preparing
    Stock Solutions
    Concentration Solvent Mass 1 mg 5 mg 10 mg
    1 mM 2.1034 mL 10.5170 mL 21.0340 mL
    5 mM 0.4207 mL 2.1034 mL 4.2068 mL
    10 mM 0.2103 mL 1.0517 mL 2.1034 mL
    *Please refer to the solubility information to select the appropriate solvent.
    In Vivo:
    • 1.

      Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

      Solubility: 2.5 mg/mL (5.26 mM); Suspended solution; Need ultrasonic

    • 2.

      Add each solvent one by one:  10% DMSO    90% corn oil

      Solubility: ≥ 2.5 mg/mL (5.26 mM); Clear solution

    *All of the co-solvents are provided by MCE.
    References
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    • Molarity Calculator

    • Dilution Calculator

    The molarity calculator equation

    Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

    Mass   Concentration   Volume   Molecular Weight *
    = × ×

    The dilution calculator equation

    Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

    This equation is commonly abbreviated as: C1V1 = C2V2

    Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
    × = ×
    C1   V1   C2   V2

    Keywords:

    Glutaminase C-IN-1Compound 968Compound968Compound-968GlutaminaseInhibitorinhibitorinhibit

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    Product Name:
    Glutaminase C-IN-1
    Cat. No.:
    HY-12682
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