Others Inhibitor

OTOP1-IN-1 (compound C2.2) is a potent zebrafish Otopetrin 1 (OTOP1) inhibitor with an IC₅₀ of 6.67 µM. OTOP1-IN-1 exhibits selectivity for zebrafish OTOP1 over mOTOP1 and hOTOP1.

Odentegravirum (Odentegravir) is a antiviral agent.

Oleanolic acid derivative 1 is an oleanolic acid derivative, which is a novel triterpenoid-steroid hybrid molecule.

Glucodichotomine B (Compound 13) is a natural product which can be isolated from the roots of Chinese medicinal plant Stellaria dichotoma L. var. lanceolata. Glucodichotomine B shows antitumor activity.

FR194738 (Standard) is the analytical standard of FR194738 (HY-100303A). This product is intended for research and analytical applications. FR194738 is a squalene epoxidase inhibitor. FR194738 inhibits squalene epoxidase activity in HepG2 cell homogenates with an IC50 of 9.8 nM.

NSC23005 (sodium) (Standard) is the analytical standard of NSC23005 (sodium) (HY-100791). This product is intended for research and analytical applications. NSC23005 sodium is a novel and effective p18 inhibitor (ED50=5.21 nM) in promoting Hematopoietic stem cells (HSCs) expansion in both murine and human models.

Lobenzarit (Standard) is the analytical standard of Lobenzarit. This product is intended for research and analytical applications. Lobenzarit, an immunomodulator, possesses anti-oxidative.

DAAO inhibitor-1 (Standard) is the analytical standard of DAAO inhibitor-1 (HY-111412). This product is intended for research and analytical applications. DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor with an IC₅₀ of 0.12 μM.

GR148672X (Standard) is the analytical standard of GR148672X (HY-110390). This product is intended for research and analytical applications. GR148672X is a triacyglycerol hydrolase (TGH) inhibitor with an IC₅₀ of 4 nM extracted from patent WO 2001016358 A2.

Trilostane (Standard) is the analytical standard of Trilostane. This product is intended for research and analytical applications. Trilostane (Win 24540) is a competitive and orally active 3-β-hydroxysteroiddehydrogenase (3β-HSD) inhibitor. Trilostane is a synthetic nonhormonal steroid. Trilostane can be used for the research of breast cancer and prostate cancer.

Ro 22-3581 (Standard) is the analytical standard of Ro 22-3581 (HY-109877). This product is intended for research and analytical applications. Ro 22-3581 (4'-(Imidazol-1-yl) acetophenone) is a selective thromboxane (Tx) synthetase inhibitor.

S-Gboxin (Standard) is the analytical standard of S-Gboxin (HY-111652). This product is intended for research and analytical applications. S-Gboxin is a functional analog of the oxidative phosphorylation (OXPHOS) inhibitor Gboxin and has antitumor activity. S-Gboxin inhibits the growth of mouse and human glioblastoma with an IC₅₀ of 470 nM. S-Gboxin has antitumor activity.

BDP-13176 (Standard) is the analytical standard of BDP-13176 (HY-111578). This product is intended for research and analytical applications. BDP-13176 is a potent fascin 1 inhibitor, with a K_d of 90 nM and an IC₅₀ of 240 nM. BDP-13176 has potential as an anti-metastatic agent.

6-O-Bis-(4,5-dimethoxy-2-nitrobenzyloxyphosphoryl)-D-trehalose is a synthetic compound that interferes with plant sugar signaling. After being absorbed by plants, 6-O-Bis-(4,5-dimethoxy-2-nitrobenzyloxyphosphoryl)-D-trehalose can trigger the release of T6P by light exposure, thereby activating the signaling pathway inside the plant. 6-O-Bis-(4,5-dimethoxy-2-nitrobenzyloxyphosphoryl)-D-trehalose can be used to study plant biosynthesis.

AS057278 (Standard) is the analytical standard of AS057278. This product is intended for research and analytical applications. AS057278 is a potent, selective, orally active and blood-brain barrier (BBB) penetrant non-peptidic D-amino acid oxidase (DAAO) inhibitor with an IC50 value of 0.91 μM and EC50 of 2.2-3.95 μM. AS057278 can normalize phencyclidine (PCP)-induced prepulse inhibition in mice. AS057278 can be used for researching schizophrenia.

CCHFV-IN-1 (compound Z10) is a potent and selective Crimean-Congo hemorrhagic fever virus (CCHFV) inhibitor. CCHFV-IN-1 exhibits potent antiviral activity (EC₅₀ = 0.60 μM) and high selectivity against CCHFV. CCHFV-IN-1 can be used for CCHFV infection research.

Voxelotor (Standard) is the analytical standard of Voxelotor. This product is intended for research and analytical applications. Voxelotor (GBT 440) is a potent inhibitor of haemoglobin S (HbS) polymerization. Voxelotor has the potential for sickle cell disease (SCD) treatment.

FR194738 free base (Standard) is the analytical standard of FR194738 free base (HY-100303). This product is intended for research and analytical applications. FR194738 free base is a squalene epoxidase inhibitor. FR194738 inhibits squalene epoxidase activity in HepG2 cell homogenates with an IC50 of 9.8 nM.

NBTGR (Standard) is the analytical standard of NBTGR (HY-108322). This product is intended for research and analytical applications. NBTGR (p-Nitrobenzylthioguanosine) is a potent inhibitor of nucleoside transport; inhibits adenosine uptake with a K_i of 70 nM.

FUBP1-IN-1 (Standard) is the analytical standard of FUBP1-IN-1 (HY-100758). This product is intended for research and analytical applications. FUBP1-IN-1 is a potent FUSE binding protein 1 (FUBP1) inhibitor which interferes with the binding of FUBP1 to its single stranded target DNA FUSE sequence , with an IC50 value of 11.0 μM.