208842-53-9
Chemical Structure
SB251023
- CAS No.: 208842-53-9
- Formula:C28H34NO6P
- Molecular Weight:511.55
IUPAC Name: ((4-((1-(((S)-2-hydroxy-3-(4-hydroxyphenoxy)propyl)amino)cyclopentyl)methyl)phenoxy)methyl)(phenyl)phosphinic acid
InChIKey: MKEFUSOCGOBQMJ-DEOSSOPVSA-N
SMILES: O=P(COC1=CC=C(C=C1)CC2(CCCC2)NC[C@@H](COC3=CC=C(C=C3)O)O)(O)C4=CC=CC=C4
Biological Activity: SB251023 is a β3-adrenergic receptor agonist with pEC50 values of 7.14 and 6.91 for the β3a- and β3b-adrenergic receptors, respectively. SB251023 is capable of modulating cyclic AMP levels and extracellular acidification rate (EAR) in cells. It has potential application value in the study of cardiovascular diseases and metabolic-related disorders[1].
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SB251023 | SB251023 is a β3-adrenergic receptor agonist with pEC50 values of 7.14 and 6.91 for the β3a- and β3b-adrenergic receptors, respectively. SB251023 is capable of modulating cyclic AMP levels and extracellular acidification rate (EAR) in cells. It has potential application value in the study of cardiovascular diseases and metabolic-related disorders. | |||||||||||||||||||||
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Keywords
