2653338-74-8

PROTAC EZH2 Degrader-38 Chemical Structure
2653338-74-8

Chemical Structure

PROTAC EZH2 Degrader-38

  • CAS No.: 2653338-74-8
  • Formula:C58H75N7O8
  • Molecular Weight:998.26

InChIKey: PDKKCVQIQSBADX-UHFFFAOYSA-N

SMILES: CCN(C1CCOCC1)C2=CC(C3=CC=C(C=C3)CN4CCN(CC4)CCCCCCCCCCCOC5=C(C6=CC=C5)C(N(C6=O)C7CCC(NC7=O)=O)=O)=CC(C(NCC8=C(C=C(NC8=O)C)C)=O)=C2C

Biological Activity: PROTAC EZH2 Degrader-38 (Compound 17) is a EZH2 PROTAC degrader with an IC50 of 165.00 nM. PROTAC EZH2 Degrader-38 functionally inhibits the methyltransferase activity of EZH2 and competitively binds to the SAM-binding pocket of the EZH2 SET domain[1].

Cat. No. Product Name Purity Description Pricing
HY-181333 		PROTAC EZH2 Degrader-38 PROTAC EZH2 Degrader-38 (Compound 17) is a EZH2 PROTAC degrader with an IC50 of 165.00 nM. PROTAC EZH2 Degrader-38 functionally inhibits the methyltransferase activity of EZH2 and competitively binds to the SAM-binding pocket of the EZH2 SET domain.
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