2. MAPK/ERK Pathway Stem Cell/Wnt
  3. ERK p38 MAPK
  4. ERK2/p38α MAPK-IN-1

ERK2/p38α MAPK-IN-1 (Compound 1, In silico Hit-2) is a potent and selective ERK2 and p38α MAPK inhibitor, with an IC50 of 82 μM for ERK2. ERK2/p38α MAPK-IN-1 binds to the allosteric site of ERK2 and p38α MAPK in distinct manners. ERK2/p38α MAPK-IN-1 can be used for the research of type 2 diabetes.

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ERK2/p38α MAPK-IN-1 構造式

ERK2/p38α MAPK-IN-1 構造式

CAS 番号 : 1016427-72-7

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ERK2/p38α MAPK-IN-1 関連抗体

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ERK アイソフォーム固有の製品をすべて表示:

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ERK ERK1 ERK2 ERK5 ERK8

p38 MAPK アイソフォーム固有の製品をすべて表示:

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p38 MAPK p38α p38β MAPK13 p38δ p38γ

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製品説明

ERK2/p38α MAPK-IN-1 (Compound 1, In silico Hit-2) is a potent and selective ERK2 and p38α MAPK inhibitor, with an IC50 of 82 μM for ERK2. ERK2/p38α MAPK-IN-1 binds to the allosteric site of ERK2 and p38α MAPK in distinct manners. ERK2/p38α MAPK-IN-1 can be used for the research of type 2 diabetes[1].

分子量

445.49

分子式

C20H16FN3O4S2
CAS 番号
SMILES

COC1=C(OC)C=C(N=C(NC(C2=CSC(COC3=CC=C(F)C=C3)=N2)=O)S4)C4=C1
輸送条件

Room temperature in continental US; may vary elsewhere.
保管条件

Please store the product under the recommended conditions in the Certificate of Analysis.
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Keywords:

ERK2/p38α MAPK-IN-11016427-72-7ERKp38 MAPKExtracellular signal regulated kinasesallosteric sitedistinct mannerstype 2 diabetesInhibitorinhibitorinhibit

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製品名:
ERK2/p38α MAPK-IN-1
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