Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal

Cat. No.: HY-152121 Purity: 95.21%: FAQs
Data Sheet SDS COA Handling Instructions

Molarity Calculator

Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal is a glucocorticoid receptor agonist. Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal can be used in anti-CD40 antibody agent conjugate (ADC). Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal can be used for the research of inflammation and immune regulation.

For research use only. We do not sell to patients.

Glucocorticoid receptor agonist-1 phosphate Ala-Ala-Mal Chemical Structure

CAS No. : 2345732-89-8

Size	Price	Stock	Quantity
1 mg	USD 450	In-stock	Estimated Time of Arrival: December 31
5 mg	USD 1450	In-stock	Estimated Time of Arrival: December 31
10 mg	USD 2400	In-stock	Estimated Time of Arrival: December 31
50 mg		Get quote
100 mg		Get quote

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Customer Review

Based on 1 publication(s) in Google Scholar

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Biological Activity
Purity & Documentation
References
Customer Review

Description

Molecular Weight

928.92

Formula

C₄₇H₅₃N₄O₁₄P

CAS No.

2345732-89-8

Appearance

Solid

Color

White to off-white

SMILES

O=P(O)(O)OCC([C@]12[C@@]3([C@@]([C@@]4([H])[C@]([C@@]5(C(CC4)=CC(C=C5)=O)C)([H])[C@H](C3)O)([H])C[C@@]1([H])O[C@@H](C6=CC=C(C=C6)CC7=CC(NC([C@H](C)NC([C@H](C)NC(CN8C(C=CC8=O)=O)=O)=O)=O)=CC=C7)O2)C)=O

Shipping

Room temperature in continental US; may vary elsewhere.

Storage

-20°C, sealed storage, away from moisture and light

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light)

Solvent & Solubility

In Vitro:

DMSO : 100 mg/mL (107.65 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)

Preparing
Stock Solutions

Concentration Solvent Mass	1 mg	5 mg	10 mg

1 mM	1.0765 mL	5.3826 mL	10.7652 mL
5 mM	0.2153 mL	1.0765 mL	2.1530 mL
10 mM	0.1077 mL	0.5383 mL	1.0765 mL

View the Complete Stock Solution Preparation Table

* Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture and light). When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.

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Dilution Calculator

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

This equation is commonly abbreviated as: C₁V₁ = C₂V₂

In Vivo Dissolution Calculator

Please enter the basic information of animal experiments:

Dosage

mg/kg

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Dosing volume
(per animal)

μL

Number of animals

Recommended: Prepare an additional quantity of animals to account for potential losses during experiments.

Calculation results:

Working solution concentration: mg/mL

Purity & Documentation

Purity: 95.21%

Select Batch:

Data Sheet (269 KB) SDS (252 KB)

COA (252 KB) HNMR (482 KB) RP-HPLC (280 KB) LCMS (99 KB)

Handling Instructions (2659 KB)

References

[1]. Adrian D. Hobson, et al. Anti-cd40 antibody drug conjugates. Patent. WO2019106608A1.

Complete Stock Solution Preparation Table

Optional Solvent	Concentration Solvent Mass	1 mg	5 mg	10 mg	25 mg

DMSO	1 mM	1.0765 mL	5.3826 mL	10.7652 mL	26.9130 mL
	5 mM	0.2153 mL	1.0765 mL	2.1530 mL	5.3826 mL
	10 mM	0.1077 mL	0.5383 mL	1.0765 mL	2.6913 mL
	15 mM	0.0718 mL	0.3588 mL	0.7177 mL	1.7942 mL
	20 mM	0.0538 mL	0.2691 mL	0.5383 mL	1.3456 mL
	25 mM	0.0431 mL	0.2153 mL	0.4306 mL	1.0765 mL
	30 mM	0.0359 mL	0.1794 mL	0.3588 mL	0.8971 mL
	40 mM	0.0269 mL	0.1346 mL	0.2691 mL	0.6728 mL
	50 mM	0.0215 mL	0.1077 mL	0.2153 mL	0.5383 mL
	60 mM	0.0179 mL	0.0897 mL	0.1794 mL	0.4485 mL
	80 mM	0.0135 mL	0.0673 mL	0.1346 mL	0.3364 mL
	100 mM	0.0108 mL	0.0538 mL	0.1077 mL	0.2691 mL