2. GPCR/G Protein Neuronal Signaling
  3. mAChR
  4. Lu 26-046

Lu 26-046 is the agonist for muscarinic M1 receptor and M2 receptor and a weak antagonist for M3 receptor, with Ki of 0.51, 26 and 5 nM, respectively. Lu 26-046 exhibits specific stimulus property, that can be recognized by rats.

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Lu 26-046

Lu 26-046 화학구조

CAS No. : 143756-51-8

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Lu 26-046 Related Antibodies

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제품 설명

Lu 26-046 is the agonist for muscarinic M1 receptor and M2 receptor and a weak antagonist for M3 receptor, with Ki of 0.51, 26 and 5 nM, respectively. Lu 26-046 exhibits specific stimulus property, that can be recognized by rats[1].

IC50 & Target

mAChR1

0.51 nM (Ki)

mAChR3

5 nM (Ki)

mAChR2

26 nM (Ki)

분자량

208.28

화학식

C10H12N2OS
CAS No.
SMILES

C#CCOC1=NSC2=C1CNC[C@H]2C
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
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Lu 26-046 Related Classifications

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Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

Keywords:

Lu 26-046143756-51-8mAChRMuscarinic acetylcholine receptorguinea-pigWistar ratInhibitorinhibitorinhibit

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상품명:
Lu 26-046
Cat. No.:
HY-120329
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