2. Others Membrane Transporter/Ion Channel Neuronal Signaling GPCR/G Protein
  3. Reference Standards GlyT 5-HT Receptor P2X Receptor
  4. Opiranserin hydrochloride (Standard)

Opiranserin hydrochloride (Standard)  (Synonyms: VVZ-149 hydrochloride (Standard))

Cat. No.: HY-109067AR
Handling Instructions Technical Support

Opiranserin hydrochloride (Standard) is the analytical standard of Opiranserin (hydrochloride) (HY-109067A). This product is intended for research and analytical applications. Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 (IC50=0.87 μM). Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain.

For research use only. We do not sell to patients.

Opiranserin hydrochloride (Standard)

Opiranserin hydrochloride (Standard) Chemical Structure

CAS No. : 1440796-75-7

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Information

Opiranserin hydrochloride (Standard) is the analytical standard of Opiranserin (hydrochloride) (HY-109067A). This product is intended for research and analytical applications. Opiranserin (VVZ-149) hydrochloride, a non-opioid and non-NSAID analgesic candidate, is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μM, respectively. Opiranserin hydrochloride shows antagonistic activity on rP2X3 (IC50=0.87 μM). Opiranserin hydrochloride is development as an injectable agent for the treatment of postoperative pain.

Application

The compound is the grade of analytical standard, which is the reference standard supplied assay. It is commonly used in qualitative, quantitative and methodological research experiments in HPLC, GC and MS.
Molecular Weight

430.97

Formula

C21H35ClN2O5
CAS No.
SMILES

O=C(C1=CC(OC)=C(OCCCC)C(OC)=C1)NCC2(CCOCC2)N(C)C.[H]Cl
Shipping

Room temperature in continental US; may vary elsewhere.
Storage

Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
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Opiranserin hydrochloride (Standard) Related Classifications

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Keywords:

Opiranserin hydrochloride (Standard)1440796-75-7VVZ-149 hydrochloride (Standard)Reference StandardsGlyT5-HT ReceptorP2X ReceptorGlycine transportersSerotonin Receptor5-hydroxytryptamine ReceptorP2XRspainanalgesicnon-opioidnon-non-steroidalanti-inflammatorypostoperativeInhibitorinhibitorinhibit

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