P2Y1/P2Y6 antagonist 1
P2Y1/P2Y6 antagonist 1 (Compound 3h) is an indolesulfonylhydrazide derivative. P2Y1/P2Y6 antagonist 1 is an orally active tP2Y1 and rP2Y6 antagonist (IC50 of 9.72 and 1.89 μM, respectively). P2Y1/P2Y6 antagonist 1 can be used in the study of neurological diseases, inflammation, cardiovascular diseases and cancer.
For research use only. We do not sell to patients.
- Formula: C17H14F3N3O4S
- Molecular Weight:413.37
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
All P2Y Receptor Isoforms
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Biological Activity
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P2Y1 Receptor 9.72 μM (IC50) |
P2Y6 Receptor 1.89 μM (IC50) |
Chemical Information
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Molecular Weight 413.37
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Formula C17H14F3N3O4S
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SMILES
O=S(C1=CC=C(OC(F)(F)F)C=C1)(NNC(CC2=CNC3=C2C=CC=C3)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)