PROTAC BRM/BRG1 degrader-1
PROTAC BRM/BRG1 degrader-1 (Example 253) is a PROTAC BRM/BRG1 degrader, with DC50 of 10-100 nM for BRM, > 1 μM for BRG1. PROTAC BRM/BRG1 degrader-1 can be used for cancer research.
(Pink: SMARCA2/BRM/BAF190B/SNF2L2 and SMARCA4/BRG1/BAF190A ligand (HY-W539427); Blue: VHL ligand (HY-168243); Black: linker (HY-168244)).
For research use only. We do not sell to patients.
- CAS No.: 2724268-88-4
- Formula: C54H63N9O9S
- Molecular Weight:1014.20
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
Biological Activity
Chemical Information
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CAS No. 2724268-88-4
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Molecular Weight 1014.20
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Formula C54H63N9O9S
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SMILES
NC(N=NC(C1=C(O)C=CC=C1)=C2)=C2OCCC3=CC=C(C(N4CC(OC5CCN(CCOC6=NOC([C@@H](C(C)C)C(N7C[C@H](O)C[C@H]7C(N[C@@H](C)C8=CC=C(C9=C(C)N=CS9)C=C8)=O)=O)=C6)CC5)C4)=O)C=C3
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
PROTAC BRM/BRG1 degrader-1 Related Classifications
HY-168242 Related Classifications
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