2. PROTAC
  3. E3 Ligase Ligand-Linker Conjugates
  4. (S,R,S,R)-AHPC-Me-CO-C7-N3

(S,R,S,R)-AHPC-Me-CO-C7-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S,R)-AHPC-Me based VHL ligand and a linker used in PROTAC technology. (S,R,S,R)-AHPC-Me-CO-C7-N3 can be connected to the ligand for protein by a linker to form PROTAC EZH2 Degrader-28 (HY-181355).

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(S,R,S,R)-AHPC-Me-CO-C7-N3

(S,R,S,R)-AHPC-Me-CO-C7-N3 화학구조

CAS No. : 2977227-44-2

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(S,R,S,R)-AHPC-Me-CO-C7-N3 Related Antibodies

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von Hippel-Lindau (VHL) MDM2 Cereblon cIAP1 Aryl Hydrocarbon Receptor TRIM21

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제품 설명

(S,R,S,R)-AHPC-Me-CO-C7-N3 is a synthesized E3 ligase ligand-linker conjugate that incorporates the (S,R,S,R)-AHPC-Me based VHL ligand and a linker used in PROTAC technology. (S,R,S,R)-AHPC-Me-CO-C7-N3 can be connected to the ligand for protein by a linker to form PROTAC EZH2 Degrader-28 (HY-181355)[1].

In Vitro

PROTACs contain two different ligands connected by a linker; one is a ligand for an E3 ubiquitin ligase and the other is for the target protein. PROTACs exploit the intracellular ubiquitin-proteasome system to selectively degrade target proteins.

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

(S,R,S,R)-AHPC-Me-CO-C7-N3 Related Antibodies
분자량

611.80

화학식

C31H45N7O4S
CAS No.
SMILES

O=C(N1[C@@H](C[C@H](C1)O)C(N[C@@H](C2=CC=C(C3=C(C)N=CS3)C=C2)C)=O)[C@H](C(C)(C)C)NC(CCCCCCCN=[N+]=[N-])=O
선적

Room temperature in continental US; may vary elsewhere.
보관

Please store the product under the recommended conditions in the Certificate of Analysis.
순도&문서
References
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(S,R,S,R)-AHPC-Me-CO-C7-N3 Related Classifications

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Keywords:

(S,R,S,R)-AHPC-Me-CO-C7-N32977227-44-2E3 Ligase Ligand-Linker ConjugatesInhibitorinhibitorinhibit

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상품명:
(S,R,S,R)-AHPC-Me-CO-C7-N3
Cat. No.:
HY-181356
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