1. Membrane Transporter/Ion Channel
    Neuronal Signaling
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  3. SDZ 220-581 Ammonium salt

SDZ 220-581 Ammonium salt 

Cat. No.: HY-13059A
Handling Instructions

SDZ 220-581 Ammonium salt is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7.

For research use only. We do not sell to patients.

SDZ 220-581 Ammonium salt Chemical Structure

SDZ 220-581 Ammonium salt Chemical Structure

CAS No. : 179411-94-0

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10 mg USD 180 In-stock
Estimated Time of Arrival: December 31
50 mg USD 768 In-stock
Estimated Time of Arrival: December 31
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Description

SDZ 220-581 Ammonium salt is an orally active, potent, competitive NMDA receptor antagonist with pKi value of 7.7[1].

IC50 & Target

pKi: 7.7 (NMDA receptor)[1]

In Vivo

SDZ 220-581 (3.2-32 mg/kg; oral administration; for 24 hours; male OF-l mice) treatment dose-dependently protects mice against maximal electroshock seizures (MES). The time-course of protection by SDZ 220-581 is characterized by a rapid onset and long duration of action[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male OF-l mice (18-26 g)[1]
Dosage: 3.2 mg/kg, 10 mg/kg, 32 mg/kg
Administration: Oral administration; for 24 hours
Result: Dose-dependently protected mice against maximal electroshock seizures (MES) upon oral administration.
Molecular Weight

386.77

Formula

C₁₆H₂₀ClN₂O₅P

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
SDZ 220-581 Ammonium salt
Cat. No.:
HY-13059A
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