1 Result for "

LML134

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "LML134" in MCE Product Catalog:

Cat. No.: HY-128656
CAS No.: 1542135-76-1
Purity:  99.43%
Target:  

Histamine Receptor

Research Areas:  

Neurological Disease Endocrinology

LML134 (compound 18b) is an orally active and high selective Histamine 3 receptor (H3R) inverse agonist with Kis of 0.3 nM and 12 nM for hH3R cAMP and hH3R bdg. LML134 penetrates the brain rapidly, leading to high H3R occupancy, and disengages its target with a fast kinetic profile. LML134 has the potential for excessive sleep disorders .
loading...
    loading...