9 Results for "

contracting guinea pig ileum

" in MedChemExpress (MCE) Product Catalog:
Products (9)

9 Results for "contracting guinea pig ileum" in MCE Product Catalog:

Cat. No.: HY-P1256C
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

JMV 449 acetate is a potent neurotensin receptor agonist. JMV 449 acetate shows an IC50 of 0.15 nM for inhibition of 125I-neurotensin binding to neonatal mouse brain and an EC50 of 1.9 nM in contracting the guinea-pig ileum. JMV 449 acetate has highly potent and long-lasting hypothermic and analgesic effects in the mouse .
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Cat. No.: HY-101222
CAS No.: 207572-69-8
Purity:  99.94%
SB-203186 hydrochloride is a potent, selective and competitive 5-HT4 antagonist. SB-203186 hydrochloride antagonizes the 5-HT4 receptor-mediated relaxations of the carbachol-contracted rat isolated oesophagus against 5-HT with pKB values of 10.9 (rat oesophagus), 9.5 (guinea-pig ileum), and 9.0 (human colon) respectively .
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Cat. No.: HY-P3895A
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Substance P (3-11) acetate is a substance P (SP) fragment peptide that can cross the BBB. Substance P (3-11) acetate has contracting activities on guinea pig ileum. Substance P (3-11) acetate also promotes human monocyte chemotaxis .
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Cat. No.: HY-P3896
CAS No.: 53749-61-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Substance P (2-11) is a substance P (SP) fragment peptide. Substance P (2-11) has contracting activities on guinea pig ileum. Substance P (2-11) inhibits the permeation of 3H SP in BBMEC monolayers .
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Cat. No.: HY-P3895
CAS No.: 51165-11-8
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Substance P (3-11) is a substance P (SP) fragment peptide that can cross the BBB. Substance P (3-11) has contracting activities on guinea pig ileum. Substance P (3-11) also promotes human monocyte chemotaxis .
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Cat. No.: HY-P1256
CAS No.: 139026-66-7
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease

JMV 449 is a potent neurotensin receptor agonist. JMV 449 shows an IC50 of 0.15 nM for inhibition of [ 125I]-neurotensin binding to neonatal mouse brain and an EC50 of 1.9 nM in contracting the guinea-pig ileum. JMV 449 has highly potent and long-lasting hypothermic and analgesic effects in the mouse .
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Cat. No.: HY-113465A
CAS No.: 75715-88-7
11-trans Leukotriene E4 is an isomer of Leukotriene E4 (LTE4). Slow isomerization of the C-11 double bond of LTE4 leads to the formation of 11-trans LTE4. 11-trans Leukotriene E4 is equipotent to LTE4 in contracting guinea pig ileum .
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Cat. No.: HY-P10599
CAS No.: 103425-21-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Scyliorhinin I is a tachykinin-1 (NK-1) and tachykinin-2 (NK-2) receptor agonist with a Ki value of 0.9 nM for rat submandibular gland NK-1 receptor and 2 nM for hamster bladder NK-2 receptor. Scyliorhinin I has the ability to contract the longitudinal muscles of the guinea pig ileum .
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Cat. No.: HY-P3809
CAS No.: 77275-70-8
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

[D-Pro2,D-Phe7,D-Trp9] Substance P is a Substance P (HY-P0201) analogue. [D-Pro2,D-Phe7,D-Trp9] Substance P is an inhibitor of Substance P. [D-Pro2,D-Phe7,D-Trp9] Substance P contracts guinea-pig ileum (GPI) indirectly .
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