35 Results for "

tachykinin NK1

" in MedChemExpress (MCE) Product Catalog:
Products (35)

35 Results for "tachykinin NK1" in MCE Product Catalog:

1
1 Cited Publications
Cat. No.: HY-151413
CAS No.: 126050-12-2
Purity:  99.69%
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

MEN 10207 is a selective NK-2 tachykinin receptor (Neurokinin Receptor) antagonist. MEN 10207 has pA2 values of 5.2, 7.9 and 4.9 in three monoreceptor in vitro assays for NK-1, NK-2 and NK-3 tachykinin receptors, respectively.
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Cat. No.: HY-P1192
CAS No.: 133156-06-6
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

GR-73632 is a tachykinin NK1 receptor agonist. GR-73632 activates spinal NK1 receptors to induce scratching, biting and licking behaviors. GR-73632 activates peripheral NK1 receptors to trigger lacrimation in guinea pigs, and activates central NK1 receptors to induce repetitive hind paw tapping behavior in gerbils. GR-73632 is applicable to research related to pruritus .
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Cat. No.: HY-P1012
CAS No.: 110880-55-2
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease Endocrinology

[Sar9,Met(O2)11]-Substance P is a tachykinin NK1 receptor selective agonist.
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Cat. No.: HY-P3092
CAS No.: 26145-48-2
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Phyllomedusin, an tachykinin decapeptide, is a NK1 receptor agonist. Phyllomedusin has vasodilating activity and provokes the contraction of the pylorus .
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Cat. No.: HY-P1193
CAS No.: 129623-01-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

GR 82334 is a potent and specific reversible tachykinin NK1 receptor antagonist . GR 82334 inhibits substance P-induced sensitization by blocking SP NK1 receptors in naked mole-rats .
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Cat. No.: HY-P3890A
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Substance P (5-11) TFA TFA, the C-terminal heptapeptide of Substance P (HY-P0201), is a neuropeptide. Substance P (5-11) TFA TFA binds to NK-1 tachykinin receptor .
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Cat. No.: HY-108479
CAS No.: 153050-21-6
Synonyms: SR140333
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Nolpitantium (SR140333) is a potent, selective, competitive, non-peptide tachykinin NK1 receptor antagonist. Nolpitantium blocks the activation of rat thalamic neurons after nociceptive stimulation .
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Cat. No.: HY-P11312
CAS No.: 2770688-17-8
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

[S5K, F6Y, L9mL, M10Mox] neurokinin A (4-10) is a neuropeptide A analog and a peptide fragment of EB1002 (HY-P10746). [S5K, F6Y, L9mL, M10Mox] neurokinin A (4-10) is highly selective for mouse tachykinin receptors and human tachykinin receptor NK1R .
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Cat. No.: HY-P10599
CAS No.: 103425-21-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Scyliorhinin I is a tachykinin-1 (NK-1) and tachykinin-2 (NK-2) receptor agonist with a Ki value of 0.9 nM for rat submandibular gland NK-1 receptor and 2 nM for hamster bladder NK-2 receptor. Scyliorhinin I has the ability to contract the longitudinal muscles of the guinea pig ileum .
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Cat. No.: HY-U00207
CAS No.: 214487-46-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease Endocrinology

MEN11467 is a selective and orally- effective peptidomimetic tachykinin NK1 receptor antagonist.
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Cat. No.: HY-P2475
CAS No.: 104486-69-3
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

[Pro9]-Substance P is a potent, reversible and selective agonist of NK-1 tachykinin receptors with an EC50 of 0.93 nM .
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Cat. No.: HY-P1379
CAS No.: 1423381-12-7
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

C14TKL-1 is a tachykinin-like peptide and exhibits an agonistic activity for neurokinin receptor 1 (NK-1) .
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Cat. No.: HY-P3890
CAS No.: 51165-09-4
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Substance P (5-11), the C-terminal heptapeptide of Substance P (HY-P0201), is a neuropeptide. Substance P (5-11) binds to NK-1 tachykinin receptor .
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Cat. No.: HY-P3889
CAS No.: 51165-07-2
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Substance P (6-11) is the C-terminal hexapeptideamide of Substance P (HY-P0201). Substance P (6-11) binds to NK-1 tachykinin receptor. Substance P (6-11) shows depolarization of motoneurons and a hypotensive effect .
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Cat. No.: HY-P1198
CAS No.: 491851-53-7
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

Hemokinin 1, human is a selective tachykinin neurokinin 1 (NK1) receptor full agonist. Hemokinin 1, human is a full agonist at NK2 and NK3 receptor. Hemokinin 1, human can produces an opioid-independent analgesia .
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Cat. No.: HY-P10619
CAS No.: 145194-26-9
Target:  

Neurokinin Receptor

Research Areas:  

Inflammation/Immunology

[Tyr6,D-Phe7,D-His9]-Substance P (6-11) is a tachykinin NK1 receptor antagonist that antagonizes Histamine (HY-B1204) induced hyperalgesia .
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Cat. No.: HY-12144
CAS No.: 136982-36-0
Research Areas:  

Neurological Disease

CP-99994 is a Tachykinin neurokinin 1 (NK-1) receptor antagonist with a Ki of 0.25 nM. CP-99994 prevents colorectal sensitization in the context of visceral hypersensitivity. CP-99994 reduces colorectal hypersensitivity induced by acetic acid injections in a model of bladder-colon cross-sensitization. CP-99994 hydrochloride attenuates the neuroglial interactions and MAPK-p38 phosphorylation associated with visceral hypersensitivity .
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Cat. No.: HY-P0255
CAS No.: 2507-24-6
Physalaemin, a non-mammalian tachykinin, binds selectively to neurokinin-1 (NK1) receptor with high affinity.
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Cat. No.: HY-119005A
CAS No.: 476494-44-7
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

YM-49598 iodide is a tachykinin NK-1 receptor antagonist. YM-49598 iodide can inhibit drug-induced bladder contraction in rats, with IC50 of 11 μg/kg .
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Cat. No.: HY-P1012A
CAS No.: 2828433-10-7
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease Endocrinology

[Sar9,Met(O2)11]-Substance P TFA is a tachykinin NK1 receptor selective agonist.
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