5-HT2CR agonist 1

5-HT2CR agonist 1 (compound 8), a 7-chloro analogue, is a selective 5-HT2CR partial agonist (Emax=71.09%) with an EC50 value of 121.5 nM and no observed activity toward 5-HT2AR or 5-HT2BR. 5-HT2CR agonist 1 exhibits no recruitment activity for β-arrestin and shows low inhibition of hERG at 10 μM.

For research use only. We do not sell to patients.

  • CAS No.: 1216074-15-5
  • Formula: C13H14ClNO
  • Molecular Weight:235.71
  • Storage:

    Please store the product under the recommended conditions in the Certificate of Analysis.

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