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  3. BEBT-908

BEBT-908 (Synonyms: PI3Kα inhibitor 1)

Cat. No.: HY-19763 Purity: >98.0%
Handling Instructions

BEBT-908 is a selective PI3Kα inhibitor extracted from patent US/20120088764A1, Compound 243, has an IC50<0.1 μM, PI3Kα inhibitor 1 also inhibits HDAC (0.1 μM≤IC50≤1 μM) .

For research use only. We do not sell to patients.

BEBT-908 Chemical Structure

BEBT-908 Chemical Structure

CAS No. : 1235449-52-1

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 469 In-stock
Estimated Time of Arrival: December 31
5 mg USD 420 In-stock
Estimated Time of Arrival: December 31
10 mg USD 600 In-stock
Estimated Time of Arrival: December 31
50 mg USD 1800 In-stock
Estimated Time of Arrival: December 31
100 mg USD 2520 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

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Customer Review

Based on 1 publication(s) in Google Scholar

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Description

BEBT-908 is a selective PI3Kα inhibitor extracted from patent US/20120088764A1, Compound 243, has an IC50<0.1 μM, PI3Kα inhibitor 1 also inhibits HDAC (0.1 μM≤IC50≤1 μM) .

IC50 & Target[1]

PI3Kα

0.1 μM (IC50)

HDAC

0.1 μM (IC50)

Molecular Weight

507.57

Formula

C₂₃H₂₅N₉O₃S

CAS No.

1235449-52-1

SMILES

CN(CC1=CC(N=C(C2=CN=C(NC)C=C2)N=C3N4CCOCC4)=C3S1)C5=NC=C(C(NO)=O)C=N5

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : ≥ 37 mg/mL (72.90 mM)

*"≥" means soluble, but saturation unknown.

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 1.9702 mL 9.8509 mL 19.7017 mL
5 mM 0.3940 mL 1.9702 mL 3.9403 mL
10 mM 0.1970 mL 0.9851 mL 1.9702 mL
*Please refer to the solubility information to select the appropriate solvent.
References
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Product Name:
BEBT-908
Cat. No.:
HY-19763
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