1. PI3K/Akt/mTOR
  2. PI3K

PI3Kα inhibitor 1 

Cat. No.: HY-19763
Handling Instructions

PI3Kα inhibitor 1 is a selective PI3Kα inhibitor extracted from patent US/20120088764A1, Compound 243, has an IC50<0.1 μM, PI3Kα inhibitor 1 also inhibits HDAC (0.1 μM≤IC50≤1 μM) .

For research use only. We do not sell to patients.
PI3Kα inhibitor 1 Chemical Structure

PI3Kα inhibitor 1 Chemical Structure

CAS No. : 1235449-52-1

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 469 In-stock
5 mg USD 420 In-stock
10 mg USD 600 In-stock
50 mg USD 1800 In-stock
100 mg USD 2520 In-stock
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

  • Biological Activity

  • Protocol

  • Technical Information

  • Purity & Documentation

  • References

Description

PI3Kα inhibitor 1 is a selective PI3Kα inhibitor extracted from patent US/20120088764A1, Compound 243, has an IC50<0.1 μM, PI3Kα inhibitor 1 also inhibits HDAC (0.1 μM≤IC50≤1 μM) .

IC50 & Target[1]

PI3Kα

0.1 μM (IC50)

HDAC

0.1 μM (IC50)

References
Preparing Stock Solutions
Concentration Volume Mass 1 mg 5 mg 10 mg
1 mM 1.9702 mL 9.8509 mL 19.7017 mL
5 mM 0.3940 mL 1.9702 mL 3.9403 mL
10 mM 0.1970 mL 0.9851 mL 1.9702 mL
Please refer to the solubility information to select the appropriate solvent.
References
Molecular Weight

507.57

Formula

C₂₃H₂₅N₉O₃S

CAS No.

1235449-52-1

SMILES

CN(CC1=CC(N=C(C2=CN=C(NC)C=C2)N=C3N4CCOCC4)=C3S1)C5=NC=C(C(NO)=O)C=N5

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Shipping

Room temperature in continental US; may vary elsewhere

Solvent & Solubility

DMSO: ≥ 37 mg/mL

* "<1 mg/mL" means slightly soluble or insoluble. "≥" means soluble, but saturation unknown.

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Product Name:
PI3Kα inhibitor 1
Cat. No.:
HY-19763
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