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GHSR Related Products (69)
Related Products (69)
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Anamorelin (Standard)
0 ImagesSynonyms: RC-1291 (Standard); ONO-7643 (Standard)Anamorelin (Standard) (RC-1291 (Standard)) is the analytical standard of Anamorelin (HY-14734). This product is intended for research and analytical applications. Anamorelin (RC-1291) is an orally active Ghrelin receptor agonist with an EC50 of 0.74 nM. Anamorelin can promote appetite, increase body weight, and stimulate the secretion of growth hormone and insulin-like growth factor-1. Anamorelin can be used in the research of anorexia and cancer cachexia.
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L-692429 hydrochloride
0 ImagesCat. No.: HY-10957ACAS No.: 169188-19-6Synonyms: MK-0751 hydrochlorideL-692429 (MK-0751) hydrochloride is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) agonist. L-692429 hydrochloride binds to G protein-coupled receptor with a Ki of 63 nM.
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GSK894281
0 ImagesCat. No.: HY-111232CAS No.: 874958-63-1GSK894281 is an orally active and highly potent ghrelin receptor full agonist with a pEC50 of <4.9 at the human motilin receptor. GSK894281 effectively enters the CNS. GSK894281 has the potential for constipation or to assist in emptying the colon prior to colonoscopy or colon surgery research.
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JMV 3002
0 ImagesCat. No.: HY-129207CAS No.: 925239-03-8Ghrelin is an endogenous ligand for the growth hormone secretagogue receptor that stimulates food intake and transduces signals to hypothalamic regulatory nuclei that control energy homeostasis. JMV3002 is a potent ghrelin receptor antagonist with an IC50 value of 1.1 nM in vitro. 80 μg/kg, JMV3002 inhibits hexarelin-stimulated food intake by as much as 98% in rats. JMV3002 alone does not elicit growth hormone release nor does it inhibit hexarelin-stimulated growth hormone secretion when tested in infant rats at a dose of 160 μg/kg.
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L-692429 (Standard)
0 ImagesCat. No.: HY-10957RCAS No.: 145455-23-8Synonyms: MK-0751 (Standard)L-692429 (Standard) is the analytical standard of L-692429 (HY-10957). This product is intended for research and analytical applications. L-692429 (MK-0751) is a benzolactam derivative and a nonpeptidyl growth hormone secretagogue (GHS) agonist. L-692429 binds to G protein-coupled receptor with a Ki of 63 nM.
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Anamorelin Fumarate
0 ImagesCat. No.: HY-14734BCAS No.: 339539-92-3Synonyms: RC-1291 Fumarate; ONO-7643 FumarateAnamorelin (RC-1291) Fumarate is an orally active Ghrelin receptor agonist with an EC50 of 0.74 nM. Anamorelin Fumarate can promote appetite, increase body weight, and stimulate the secretion of growth hormone and insulin-like growth factor-1. Anamorelin Fumarate can be used in the research of anorexia and cancer cachexia.
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Ghrelin receptor full agonist-3
0 ImagesCat. No.: HY-180210CAS No.: 2243167-93-1Ghrelin receptor full agonist-3 (Compound 22) is a selective, potent and orally active ghrelin receptor full agonist with an EC50 of 1.8 nM. Ghrelin receptor full agonist-3 can stimulate pulsatile secretion of growth hormone (GH), significantly increasing the frequency and duration of GH secretion, thereby inducing a sustained increase in insulin-like growth factor-1 (IGF-1) levels. Ghrelin receptor full agonist-3 can be used for the researches of cancer and chronic obstructive pulmonary disease.
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SM-130686
0 ImagesCat. No.: HY-116959CAS No.: 259667-25-9SM-130686 is an oxindole derivative and an active GH secretagogue (GHS). SM-130686 stimulates GH release with a Half-maximum stimulation of 6.3 nM. SM-130686 has an orally active.
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KwFwLL-NH2
0 ImagesCat. No.: HY-P10673CAS No.: 942266-38-8KwFwLL-NH2, a hexapeptide, is a ghrelin receptor ligand. KwFwLL-NH2 can act as a specific inverse agonist at the ghrelin receptor but with moderate potency (EC50=45.6 nM).
