116644-53-2
116644-53-2
Chemical Structure
Mibefradil
Synonym(s): Ro 40-5967
- CAS No.: 116644-53-2
- Formula:C29H38FN3O3
- Molecular Weight:495.63
IUPAC Name: (1S,2S)-2-(2-((3-(1H-benzo[d]imidazol-2-yl)propyl)(methyl)amino)ethyl)-6-fluoro-1-isopropyl-1,2,3,4-tetrahydronaphthalen-2-yl 2-methoxyacetate
InChIKey: HBNPJJILLOYFJU-VMPREFPWSA-N
SMILES: O=C(O[C@@]1(CCN(CCCC2=NC3=CC=CC=C3N2)C)[C@@H](C(C)C)C4=C(C=C(F)C=C4)CC1)COC
Biological Activity: Mibefradil (Ro 40-5967) is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels displaying IC50s of 2.7 μM and 18.6 μM for T-type and L-type currents, respectively[1].
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Mibefradil | Mibefradil (Ro 40-5967) is a calcium channel blocker with moderate selectivity for T-type Ca2+ channels displaying IC50s of 2.7 μM and 18.6 μM for T-type and L-type currents, respectively. | |||||||||||||||||||||
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References
Keywords
