125989-15-3
Chemical Structure
L-659874
- CAS No.: 125989-15-3
- Formula:C40H55N9O8S
- Molecular Weight:822.00
IUPAC Name: (S)-2-((S)-2-((S)-2-acetamido-4-methylpentanamido)-4-(methylthio)butanamido)-N1-((S)-1-(((S)-1-((2-amino-2-oxoethyl)amino)-1-oxo-3-phenylpropan-2-yl)amino)-3-(1H-indol-3-yl)-1-oxopropan-2-yl)pentanediamide
InChIKey: RDESGNZZHYRWNM-ZTTXAYQISA-N
SMILES: C([C@@H](C(N[C@@H](CC1=CC=CC=C1)C(NCC(N)=O)=O)=O)NC([C@@H](NC([C@@H](NC([C@H](CC(C)C)NC(C)=O)=O)CCSC)=O)CCC(N)=O)=O)C=2C=3C(NC2)=CC=CC3
Biological Activity: L-659874 is a selective NK2 receptor antagonist with an IC50 value of 0.49 μM in hamsters. L-659874 inhibits NK2 receptor-mediated hydrolysis of inositol phospholipids. L-659874 could be used for research on the correlation between pain signal transduction and smooth muscle responses[1].
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L-659874 | L-659874 is a selective NK2 receptor antagonist with an IC50 value of 0.49 μM in hamsters. L-659874 inhibits NK2 receptor-mediated hydrolysis of inositol phospholipids. L-659874 could be used for research on the correlation between pain signal transduction and smooth muscle responses. | |||||||||||||||||||||
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