2488867-43-0
2488867-43-0
Chemical Structure
P300-IN-2
- CAS No.: 2488867-43-0
- Formula:C26H27FN4O5
- Molecular Weight:494.52
IUPAC Name: 1-((R)-3'-(2-((2R,5R)-2-(4-fluorophenyl)-5-methylpyrrolidin-1-yl)-2-oxoethyl)-2',4'-dioxo-2,3-dihydrospiro[indene-1,5'-oxazolidin]-5-yl)-3-methylurea
InChIKey: RGUSDFBEDZBTQP-MDGPWXEQSA-N
SMILES: O=C1[C@@]2(C=3C(CC2)=CC(NC(NC)=O)=CC3)OC(=O)N1CC(=O)N4[C@H](CC[C@H]4C)C5=CC=C(F)C=C5
Biological Activity: P300-IN-2 is a p300 inhibitor (IC50=3.6 μM) that inhibits histone acetyltransferase p300 activity. P300-IN-2 shows weak inhibitory activity against CWR22RV1 cell proliferation. P300-IN-2 can be used for research on p300-mediated diseases, such as cancer[1].
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P300-IN-2 | P300-IN-2 is a p300 inhibitor (IC50=3.6 μM) that inhibits histone acetyltransferase p300 activity. P300-IN-2 shows weak inhibitory activity against CWR22RV1 cell proliferation. P300-IN-2 can be used for research on p300-mediated diseases, such as cancer. | |||||||||||||||||||||
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