2815263-05-7
2815263-05-7
Chemical Structure
GPR84 antagonist 3
- CAS No.: 2815263-05-7
- Formula:C29H27N5O
- Molecular Weight:461.56
IUPAC Name: 4-(4-(3-((1H-indol-3-yl)methyl)-5-phenyl-1,2,4-triazin-6-yl)benzyl)morpholine
InChIKey: XGBKJLWLVCHTCR-UHFFFAOYSA-N
SMILES: N1(CC2=CC=C(C3=C(C4=CC=CC=C4)N=C(CC5=CNC6=C5C=CC=C6)N=N3)C=C2)CCOCC1
Biological Activity: GPR84 antagonist 3 (compound 42) is a potent GPR84 (G-protein-coupled receptor 84) antagonist. GPR84 antagonist 3 inhibits GTPγS, with a pIC50 of 8.28. GPR84 antagonist 3 has a favorable pharmacokinetic profile suitable[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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GPR84 antagonist 3 | 98.32% | GPR84 antagonist 3 (compound 42) is a potent GPR84 (G-protein-coupled receptor 84) antagonist. GPR84 antagonist 3 inhibits GTPγS, with a pIC50 of 8.28. GPR84 antagonist 3 has a favorable pharmacokinetic profile suitable. | ||||||||||||||||||||
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