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Referencia número: HY-123447

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GR-175737

GR 175737 is a partial histamine H3 receptor agonist, with an EC₅₀ of 7.8 nM. GR 175737 can be used in the research of inflammatory diseases.

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No. CAS: 176860-26-7
Fòrmula: C₁₄H₁₃ClN₄O
Peso molecular:288.73

Almacenamiento:

Please store the product under the recommended conditions in the Certificate of Analysis.

Data Sheet (266 KB)

GR-175737 Chemical Structure

No. CAS: 176860-26-7

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Actividad biológica

Descripciòn

GR 175737 is a partial histamine H3 receptor agonist, with an EC₅₀ of 7.8 nM. GR 175737 can be used in the research of inflammatory diseases^[1].

IC₅₀ & Target^[1]

H₃ receptor

7.8 nM (EC₅₀)

Ver todos los productos específicos de isoformas Histamine Receptor :

Chemical Information

No. CAS 176860-26-7
Peso molecular 288.73
Fòrmula C₁₄H₁₃ClN₄O
SMILES

ClC1=CC=C(C=C1)CC2=NOC(CCC3=CN=CN3)=N2
Envío

Room temperature in continental US; may vary elsewhere.
Almacenamiento

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureza y Documentación

Select Batch:

Pureza: 99.98%

Assay: 99.98%

ee.: 99.98%

Ficha de datos (266 KB)
COA (2659 KB)
Elemental Analysis Report (2659 KB)
HNMR (2659 KB)
CNMR (2659 KB)
RP-HPLC (2659 KB)
NP-HPLC (2659 KB)
MS (2659 KB)
LCMS (2659 KB)
IR (2659 KB)
GC (2659 KB)
OR (2659 KB)
SDS-PAGE (2659 KB)
SEC-HPLC (2659 KB)
Other Report (2659 KB)
Instrucciones de manejo (2659 KB)

Referencias

[1]. Soudijn W, et al. Structure–activity relationships of inverse agonists for G‐protein‐coupled receptors. Medicinal research reviews, 2005, 25(4): 398-426.

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Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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100 mg

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GR-175737

Ver todos los productos específicos de isoformas Histamine Receptor

Actividad biológica

Chemical Information

Pureza y Documentación

Referencias

Calculators

Help & FAQs

GR-175737 Related Classifications

HY-123447 Related Classifications