Glasdegib maleate
Based on 5 publication(s) in Google Scholar
Glasdegib maleate (PF-04449913 maleate) is a potent and orally bioavailable smoothened inhibitor. Glasdegib maleate binds to human SMO (amino acids 181-787) with IC50value of 4 nM.
For research use only. We do not sell to patients.
- CAS No.: 2030410-25-2
- Formula: C25H26N6O5
- Molecular Weight:490.51
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Biological Activity
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Chemical Information
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Publications Citing Use of MedChemExpress (MCE) Glasdegib maleate
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Biological Activity
Chemical Information
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CAS No. 2030410-25-2
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Molecular Weight 490.51
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Formula C25H26N6O5
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SMILES
O=C(NC1=CC=C(C#N)C=C1)N[C@H]2C[C@H](C3=NC4=CC=CC=C4N3)N(C)CC2.OC(/C=C\C(O)=O)=O
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Synonyms
PF-04449913 maleate
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Publications (5)
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Journal Impact Factor
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Most Recent
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Molecules
Development and Validation of a Rapid LC-MS/MS Method for Quantifying Alvocidib: In Silico and In Vitro Metabolic Stability Estimation in Human Liver Microsomes. [Abstract]2023 Mar 4;28(5):2368. PMID: 36903615 -
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Methods Mol Biol
2018:1711:351-398. PMID: 29344898
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Glasdegib maleate Related Classifications
HY-16391A Related Classifications
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