RP 73163 Racemate
RP 73163 Racemate is the racemate of RP 73163. RP 73163 is a potent ACAT inhibitor, with cholesterol lowering activity.
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研究用途以外に使用した場合、当社は一切の責任を負いかねます。
- CAS 番号: 136609-53-5
- 分子式: C25H28N4OS
- 分子量:432.58
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
生物活性
製品説明
Cellular Effect
|
Cell Line
|
Type | Value | Description | References |
|---|---|---|---|---|
| HepG2 | IC50 |
108 nM
Compound: 5
|
Compound was evaluated for inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase in microsomes from HEP G2 cells.
Compound was evaluated for inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase in microsomes from HEP G2 cells.
|
10.1016/0960-894X(95)00555-8 |
| THP-1 | IC50 |
164 nM
Compound: 5
|
Compound was evaluated for inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase in microsomes from THP-1 cells.
Compound was evaluated for inhibitory activity against Acyl coenzyme A:cholesterol acyltransferase in microsomes from THP-1 cells.
|
10.1016/0960-894X(95)00555-8 |
化学情報
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CAS 番号 136609-53-5
-
分子量 432.58
-
分子式 C25H28N4OS
-
SMILES
CC1=CC(C)=NN1CCCCCS(C2=NC(C3=CC=CC=C3)=C(C4=CC=CC=C4)N2)=O
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輸送条件
Room temperature in continental US; may vary elsewhere.
-
保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)