(+)-Eseroline
(+)-Eseroline is an opioid agonist and adenylate cyclase inhibitor (Ki=6-8 μM). (+)-Eseroline binds specifically to μ-opioid receptors and δ-opioid receptors on rat brain cell membranes (Ka=0.7 μM). (+)-Eseroline exhibits only weak activity in various mouse analgesic models and can be used for studies on pain-related mechanisms.
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- CAS 番号: 29347-15-7
- 分子式: C13H18N2O
- 分子量:218.30
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保管条件:
Please store the product under the recommended conditions in the Certificate of Analysis.
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生物活性
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化学情報
- 純度とドキュメンテーション
- 参考文献
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Opioid Receptor アイソフォーム固有の製品をすべて表示
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生物活性
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μ Opioid Receptor/MOR |
δ Opioid Receptor/DOR |
(+)-Eseroline (0-100 μM; 10 min) inhibits adenylate cyclase activity in NG108-15 cell membranes with a Ki of 6-8 μM, acts as a lower-efficacy opiate agonist relative to (-)-Eseroline, and functions as an antagonist of both (-)-Eseroline and the opioid peptide dalamid[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.
化学情報
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CAS 番号 29347-15-7
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分子量 218.30
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分子式 C13H18N2O
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SMILES
C[C@@]12C=3C(N(C)[C@@]1(N(C)CC2)[H])=CC=C(O)C3
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輸送条件
Room temperature in continental US; may vary elsewhere.
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保管条件
Please store the product under the recommended conditions in the Certificate of Analysis.
純度とドキュメンテーション
参考文献
Calculators
濃度 (開始) × 体積 (開始) = 濃度 (終了) × 体積 (終了)
(+)-Eseroline 関連分類
HY-W387210 関連分類
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