29347-15-7
Chemical Structure
(+)-Eseroline
- CAS No.: 29347-15-7
- Formula:C13H18N2O
- Molecular Weight:218.30
IUPAC Name: (3aR,8aS)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydropyrrolo[2,3-b]indol-5-ol
InChIKey: HKGWQUVGHPDEBZ-QWHCGFSZSA-N
SMILES: C[C@@]12C=3C(N(C)[C@@]1(N(C)CC2)[H])=CC=C(O)C3
Biological Activity: (+)-Eseroline is an opioid agonist and adenylate cyclase inhibitor (Ki=6-8 μM). (+)-Eseroline binds specifically to μ-opioid receptors and δ-opioid receptors on rat brain cell membranes (Ka=0.7 μM). (+)-Eseroline exhibits only weak activity in various mouse analgesic models and can be used for studies on pain-related mechanisms[1].
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(+)-Eseroline | (+)-Eseroline is an opioid agonist and adenylate cyclase inhibitor (Ki=6-8 μM). (+)-Eseroline binds specifically to μ-opioid receptors and δ-opioid receptors on rat brain cell membranes (Ka=0.7 μM). (+)-Eseroline exhibits only weak activity in various mouse analgesic models and can be used for studies on pain-related mechanisms. | |||||||||||||||||||||
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Keywords
