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Kgp-IN-1 hydrochloride 

Cat. No.: HY-128523A Purity: 95.52%
Handling Instructions

Kgp-IN-1 hydrochloride is an arginine-specific gingipain (Rgp) inhibitor extracted from patent WO2017201322A1, compound 13-R.

For research use only. We do not sell to patients.

Kgp-IN-1 hydrochloride Chemical Structure

Kgp-IN-1 hydrochloride Chemical Structure

CAS No. : 2097865-47-7

Size Price Stock Quantity
10 mM * 1  mL in DMSO USD 450 In-stock
Estimated Time of Arrival: December 31
5 mg USD 450 In-stock
Estimated Time of Arrival: December 31
10 mg USD 780 In-stock
Estimated Time of Arrival: December 31
50 mg USD 2300 In-stock
Estimated Time of Arrival: December 31
100 mg USD 3600 In-stock
Estimated Time of Arrival: December 31
200 mg   Get quote  
500 mg   Get quote  

* Please select Quantity before adding items.

Customer Review

Based on 1 publication(s) in Google Scholar

Other Forms of Kgp-IN-1 hydrochloride:

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Description

Kgp-IN-1 hydrochloride is an arginine-specific gingipain (Rgp) inhibitor extracted from patent WO2017201322A1, compound 13-R[1].

IC50 & Target

Rgp[1]

Molecular Weight

468.87

Formula

C₁₉H₂₅ClF₄N₄O₃

CAS No.

2097865-47-7

SMILES

O=C(N[[email protected]@H](CCCNC(N)=N)C(COC1=C(F)C(F)=CC(F)=C1F)=O)C2CCCC2.Cl

Shipping

Room temperature in continental US; may vary elsewhere.

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
Solvent & Solubility
In Vitro: 

DMSO : 125 mg/mL (266.60 mM; Need ultrasonic)

Preparing
Stock Solutions
Concentration Solvent Mass 1 mg 5 mg 10 mg
1 mM 2.1328 mL 10.6639 mL 21.3279 mL
5 mM 0.4266 mL 2.1328 mL 4.2656 mL
10 mM 0.2133 mL 1.0664 mL 2.1328 mL
*Please refer to the solubility information to select the appropriate solvent.
In Vivo:
  • 1.

    Add each solvent one by one:  10% DMSO    40% PEG300    5% Tween-80    45% saline

    Solubility: ≥ 2.08 mg/mL (4.44 mM); Clear solution

  • 2.

    Add each solvent one by one:  10% DMSO    90% (20% SBE-β-CD in saline)

    Solubility: ≥ 2.08 mg/mL (4.44 mM); Clear solution

  • 3.

    Add each solvent one by one:  10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (4.44 mM); Clear solution

*All of the co-solvents are provided by MCE.
References
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  • Molarity Calculator

  • Dilution Calculator

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

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The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
× = ×
C1   V1   C2   V2

Keywords:

Kgp-IN-1OthersInhibitorinhibitorinhibit

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Product Name:
Kgp-IN-1 hydrochloride
Cat. No.:
HY-128523A
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