1 Result for "

mct4-in-1

" in MedChemExpress (MCE) Product Catalog:
Products (1)

1 Results for "mct4-in-1" in MCE Product Catalog:

Cat. No.: HY-132301
CAS No.: 2445185-57-7
Purity:  98.89%
Synonyms: mct4-in-1
Research Areas:  

Cancer

MSC-4381 (MCT4-IN-1), a chemical probe, is an orally active and selective monocarboxylate transporter 4 (MCT4/SLC16A3) inhibitor with an IC50 of 77 nM and a Ki of 11 nM. MSC-4381 targets to the cytosolic domain of MCT4. MSC-4381 results in lactate efflux inhibition and reduction of cellular viability in MCT4 high expressing cells. MSC-4381 has the potential for MCT4 transporter inhibition research . MSC-4381 is a click chemistry reagent, it contains an Alkyne group and can undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.