88 Results for "

G-{d-Arg}-GDSP

" in MedChemExpress (MCE) Product Catalog:
Products (88)

88 Results for "G-{d-Arg}-GDSP" in MCE Product Catalog:

Cat. No.: HY-P11405
CAS No.: 122481-75-8
Target:  

Neurotensin Receptor

Research Areas:  

Neurological Disease Cancer

[D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P is a potent inhibitor of cell growth in small cell lung cancer (SCLC). [D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P is also a neuropeptide antagonist, capable of blocking colony formation stimulated by various neuropeptides (including vasopressin and bradykinin). [D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P inhibits the mobilization of Ca 2+ and the activation of mitogen-activated protein kinases induced by vasopressin or bradykinin. [D-Arg1, D-Trp5, 7, 9, Leu11]-Substance P inhibits the growth of H-69 xenograft tumors in nude mice .
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Cat. No.: HY-P5591
Target:  

Fungal

Research Areas:  

Infection

PAF26 is an antimicrobial peptide against phytopathogenic fungi Penicillium digitatum, Penicillium italicum and Botrytis cinerea .
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Cat. No.: HY-P0041A
Target:  

Vasopressin Receptor

Research Areas:  

Neurological Disease

F992 TFA is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue .
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Cat. No.: HY-P5327
Target:  

Bcl-2 Family

Research Areas:  

Others

r8 Bid BH3 is a biological active peptide. (The Bid BH3 is a pro-apoptotic member of the 'BH3-only' subset of BCL-2 family proteins that constitute a critical control point in apoptosis. r8BIDBH3 is lethal to human leukemia cell lines that expresse Bcl-2. The Bcl-2 antagonists may have the potential to be efficacious in cancer therapy. Poly-D-arginine (d-isomer as denoted by rrrrrrrr) is fused to the Bid BH3 peptide to facilitate cellular uptake of the peptide.)
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Cat. No.: HY-P5329
Target:  

NADPH Oxidase

Research Areas:  

Others

r8-Gly-Noxa A BH3 is a biological active peptide. (This cell permeable peptide is derived from the BH3 domain (a death domain) of Noxa A, amino acid residues 17 to 36. Eight D-Arginine residues and a Glycine linker residue are added to the amino terminal of the peptide.)
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Cat. No.: HY-P10824
CAS No.: 1430219-69-4
Target:  

Amyloid-β

Research Areas:  

Neurological Disease

RI-OR2-TAT is a brain-penetrant inhibitor of β-Amyloid oligomerization, which is produced by adding the HIV protein transduction domain TAT to RI-OR2. RI-OR2-TAT binds to Aβ42 fibrils with a Kd value of 58-125 nM. RI-OR2-TAT reduces aggregation and plaque levels, reduces activation of microglia and oxidative damage, and increases the number of young neurons in the dentate gyrus .
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Cat. No.: HY-P0206F
CAS No.: 477319-71-4
Target:  

Bradykinin Receptor

Research Areas:  

Others

biotin-Bradykinin is a biological active peptide. (Biotin labeled HY-P0206)
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Cat. No.: HY-P11384
CAS No.: 144161-76-2
Target:  

Integrin

Research Areas:  

Cardiovascular Disease

D-RGDW is an Arg-Gly-Asp (RGD) containing peptide. D-RGDW inhibits αIIbβ3 mediated platelet aggregation .
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Cat. No.: HY-P4139
Target:  

Inhibitory Antibodies

Research Areas:  

Others

activable cell-penetrating peptide (ACCP) consists of a polycationic CPP (typically arg9 or r9) connected via a cleavable linker to a matching polyanion (typically glu9 or e9), which reduces the net charge to nearly zero and thereby inhibits adhesion and uptake into cells .
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Cat. No.: HY-138152
CAS No.: 113711-77-6
Synonyms: Benzyl-D-Arg-Gly-Arg-pNA dihydrochloride
Target:  

Fluorescent Dye

Research Areas:  

Others

Z-D-Arg-Gly-Arg-pNA dihydrochloride is a hydrolytic chromogenic plasmin substrate .
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Cat. No.: HY-103292
CAS No.: 118122-39-7
Target:  

Bradykinin Receptor

Research Areas:  

Cardiovascular Disease

[Phe8Ψ(CH-NH)Arg9]-Bradykinin is a selective Bradykinin receptor B2 agonist (not cleaved by protein kinase I/II). [Phe8Ψ(CH-NH)Arg9]-Bradykinin has potential for the research of hypertension .
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Cat. No.: HY-P0198B
[D-Arg25]-Neuropeptide Y (human) ([D-Arg25] NPY) is a Y1 receptor selective agonist. Neuropeptide Y (human) is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity .
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Cat. No.: HY-P3870B
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

DALDA TFA is a potent and highly selective μ-opioid receptor agonist with a Ki of 1.69 nM. DALDA TFA shows antinociceptive and respiratory effects .
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Cat. No.: HY-P4335
CAS No.: 782432-03-5
Target:  

Ser/Thr Protease

Research Areas:  

Others

Bz-RGFFP-4MβNA, a substrate for Cathepsin D, is suitable for either colorimetric or fluorometric assay .
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Cat. No.: HY-P4544
CAS No.: 1926163-57-6
Target:  

MALT1 NF-κB MMP

Research Areas:  

Cancer

Z-Val-Arg-Pro-DL-Arg-Fluoromethylketone is an irreversible MALT1 protein inhibitor. Z-Val-Arg-Pro-DL-Arg-Fluoromethylketone inhibits the growth and invasion of diffuse large B-cell lymphoma by inhibiting MALT1-induced NF-κB activation and MMP expression .
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Cat. No.: HY-P5509
CAS No.: 230968-98-6
Target:  

Inhibitory Antibodies

Research Areas:  

Others

C5aR1 antagonist peptide is a biological active peptide. (This linear peptide is derived from the C-terminus of the chemokine, complement fragment 5 anaphylatoxin (C5a). This peptide functions to inhibit C5a binding and function at human and rat C5a receptors. C5a is crucial to triggering cellular immune responses and its overexpression is involved in arthritis, Alzheimer’s disease, cystic fibrosis, systemic lupus erythematosus, and other immunoinflammatory diseases.)
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Cat. No.: HY-P10823
CAS No.: 1219627-58-3
Target:  

Amyloid-β

Research Areas:  

Neurological Disease

RI-OR2, a retro-inverso peptide, is an amyloid-β (Aβ) oligomerization inhibitor. RI-OR2 binds to immobilized β-Amyloid (1-42) (HY-P1363A) monomers and fibrils, with an apparent Kd of 9-12 μM, and also acted as an inhibitor of Aβ(1-42) fibril extension .
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Cat. No.: HY-P10930
Target:  

DNA/RNA Synthesis

Research Areas:  

Cancer

wrwyar-NH2 (TFA) is a control peptide for wrwycr-NH2 (HY-P10930A) .
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Cat. No.: HY-P10418
Target:  

c-Myc

Research Areas:  

Cancer

VGN50 is a bioactive molecule that mimics the function of K-Rta and down-regulates MYC-mediated gene transcription. VGN50 has antitumor activity .
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Cat. No.: HY-P10930A
Target:  

DNA/RNA Synthesis

Research Areas:  

Cancer

wrwycr-NH2 (TFA) is a peptide. wrwycr-NH2 (TFA) is cytotoxic to multiple cancer cells, can induce DNA damage and cell cycle arrest, but does not induce endoplasmic reticulum stress. wrwycr-NH2 (TFA) has anti-tumor activity, and it shows better efficacy when used in combination with DNA-damaging agents .
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