88 Results for "

G-{d-Arg}-GDSP

" in MedChemExpress (MCE) Product Catalog:
Products (88)

88 Results for "G-{d-Arg}-GDSP" in MCE Product Catalog:

Cat. No.: HY-P1577
CAS No.: 115814-08-9
Target:  

Opioid Receptor

Research Areas:  

Inflammation/Immunology

Dermorphin Analog is an analog of Dermorphin. Dermorphin is a natural heptapeptide μ-opioid receptor agonist found in amphibian skin.
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Cat. No.: HY-P5753A
Target:  

Bacterial

Research Areas:  

Infection

JB-95 acetate, a β-hairpin macrocyclic peptide, exhibits potent antimicrobial activity against Escherichia coli. JB-95 acetate can selectively disrupt the outer membrane but not the inner membrane of E. coli .
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Cat. No.: HY-P10922
CAS No.: 1246741-19-4
Target:  

Cathepsin

Research Areas:  

Others

Cathepsin E substrate e is a substrate of Cathepsin E. Cathepsin E substrate e was designed in such a way that due to the close proximity of a Mca-donor and a Dnp-acceptor, a near complete intramolecular quenching effect was achieved in its intact state. After the proteolytic cleavage of the hydrophobic motif of the peptide substrate, both Mca and Dnp would be further apart, resulting in bright fluorescence .
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Cat. No.: HY-P2118
CAS No.: 109333-26-8
Target:  

Bradykinin Receptor

Research Areas:  

Inflammation/Immunology

NPC-567 is a bradykinin B2 receptor antagonist. NPC-567 is effective in inhibiting the acute response to allergen in the airways .
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Cat. No.: HY-P1194A
Target:  

Neurokinin Receptor

Research Areas:  

Inflammation/Immunology

Spantide I TFA, a substance P analog, is a selective NK1 receptor antagonist, with Ki values of 230 nM and 8150 nM for NK1 and NK2 receptor, respectively. Spantide I provides an approach to reduce type 1 and enhance the type 2 cytokine IL-10 in the infected cornea, leading to a significant reduction in corneal perforation .
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Cat. No.: HY-136623
CAS No.: 88331-14-0
Target:  

Opioid Receptor

Research Areas:  

Neurological Disease

BW443C is a selective opioid receptor agonist. BW443C has antinociceptive effect .
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Cat. No.: HY-P10046
CAS No.: 64158-84-5
Target:  

Vasopressin Receptor

Research Areas:  

Metabolic Disease

[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an arginine-vasopressin (AVP) antagonist. AVP-A can significantly lower plasma aldosterone concentration in rats. AVP-A can be used for the research of the growth and steroidogenic capacity of rat adrenal zona glomerulosa .
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Cat. No.: HY-P3082
CAS No.: 126053-71-2
Target:  

Endogenous Metabolite

Research Areas:  

Cardiovascular Disease

SKF 106760 is a potent platelet fibrin receptor (glycoprotein IIb/IIIa) antagonist with significant antiplatelet and antithrombotic activities. SKF 106760 inhibits platelet aggregation in dogs in vitro and prevents thrombus formation in stenotic carotid arteries. SKF 106760 has also shown elimination effects against aspirin-resistant thrombi that develop in the setting of high-grade stenosis .
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Cat. No.: HY-P5518
CAS No.: 1054763-33-5
[Des-Arg10]-HOE I40 is a potent bradykinin B1 receptor antagonist .
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Cat. No.: HY-P1194B
Target:  

Neurokinin Receptor

Research Areas:  

Neurological Disease

[D-Pro2] Spantide I TFA is a Spantide analog. Spantide I is a selective NK1 receptor antagonist .
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Cat. No.: HY-P10118
CAS No.: 478164-48-6
Target:  

Cathepsin

Research Areas:  

Others

Cathepsin L-IN-3 (Compound cat L inh. 7) is selective a noncovalent cathepsin L inhibitor with a Ki of 4.3 nM .
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Cat. No.: HY-P3225
CAS No.: 143077-65-0
(D-Arg1,D-Pro2,D-Trp7,9,L-Leu11)-Substance P (acetate) is an antagonist for Substance P (HY-P0201) and Bombesin (HY-P0195) that has effects on ocular inflammatory responses to antidromic trigeminal nerve stimulation .
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Cat. No.: HY-103289
CAS No.: 235082-52-7
Purity:  99.15%
MEN 11270, a cyclic decapeptide, is a B2 kinin receptor antagonist. MEN 11270 bound with high-affinity to the B2 kinin receptor constitutively expressed by WI38 human fibroblasts, inhibiting 3H-bradykinin (BK) with a pKi value of 10.3 .
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Cat. No.: HY-P2028
CAS No.: 106881-54-3
Target:  

GnRH Receptor

Research Areas:  

Cancer

BIM 21009 is a LHRH and GnRH receptor antagonist. BIM 21009 inhibits tumor growth .
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Cat. No.: HY-P2446
CAS No.: 83539-08-6
Synonyms: APTAA-LHRH
Target:  

GnRH Receptor

Research Areas:  

Endocrinology

ORG 30276 (APTAA-LHRH) is a potent GnRH antagonist that effectively reduces serum LH and FSH levels in male rats. ORG 30276 significantly decreases unoccupied pituitary GnRH receptors, leading to suppressed gonadotropin secretion. ORG 30276 treatment results in a considerable reduction in mRNA levels of gonadotropin beta-subunits in the pituitary gland. ORG 30276's effects on gonadotropin dynamics can be selectively reversed by the replacement of specific sex steroids, with androgens being particularly effective for the FSH beta-subunit mRNA levels.
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Cat. No.: HY-P0041
CAS No.: 162277-99-8
Target:  

Vasopressin Receptor

Research Areas:  

Neurological Disease

F992 is an antidiuretic peptide and vasopressin (antidiuretic hormone) analogue .
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Cat. No.: HY-P11668
CAS No.: 2650595-42-7
Target:  

CaSR

Research Areas:  

Neurological Disease

Gosicalcetide is a calcium sensing receptor (CaSR) agonist .
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Cat. No.: HY-P11894
Target:  

Bacterial

Research Areas:  

Infection

Antimicrobial peptide 6b is a cationic macrocyclic antimicrobial peptide. It exhibits broad-spectrum antibacterial and antifungal activities, with a MIC of 1.5-6.2 μg/mL against drug-resistant Gram-positive bacteria, a MIC of 4-25 μg/mL against Gram-negative bacteria, and also shows activity against pathogenic fungi. It acts through a membrane disruption mechanism, has a unique "sandwich" conformation, low hemolytic activity, and can rapidly kill bacteria and eliminate bacterial and fungal biofilms. Antimicrobial peptide 6b can be used in studies of drug-resistant bacterial infections and fungal infections .
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Cat. No.: HY-P11832
CAS No.: 3057162-39-4
Target:  

CaSR

Research Areas:  

Endocrinology

CaSR agonist peptide-1 is a human calcium-sensing receptor (CaSR) agonist. CaSR agonist peptide-1 activates CaSR by binding to it. CaSR agonist peptide-1 can be used in studies related to secondary hyperparathyroidism .
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