57 Results for "

β-Lactamase-IN-1

" in MedChemExpress (MCE) Product Catalog:
Products (57)

57 Results for "β-Lactamase-IN-1" in MCE Product Catalog:

Cat. No.: HY-19773
CAS No.: 1075237-97-6
Research Areas:  

Infection

β-Lactamase-IN-1 is an inhibitor of β-Lactamase extracted from patent WO2016027249A1, page 77. β-Lactamase-IN-1 can be used to prepare of tricyclic nitrogen containing compound. β-Lactamase-IN-1 can be used for the research of neisseria gonorrhea infection [1].
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95
95 Publications Verification
Cat. No.: HY-14879A
CAS No.: 1192491-61-4
Purity:  99.99%
Synonyms: NXL-104; AVE1330A
Research Areas:  

Infection

Avibactam sodium (NXL-104) is a covalent and reversible non-β-lactam β-lactamase inhibitor which inhibits β-lactamase TEM-1 and CTX-M-15 with IC50s of 8 nM and 5 nM, respectively [1].
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95
95 Publications Verification
Cat. No.: HY-14879
CAS No.: 1192500-31-4
Purity:  99.22%
Synonyms: NXL-104 free acid; AVE1330A free acid
Research Areas:  

Infection

Avibactam (NXL-104) free acid is a covalent and reversible non-β-lactam β-lactamase inhibitor which inhibits β-lactamase TEM-1 and CTX-M-15 with IC50s of 8 nM and 5 nM, respectively [1].
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95
95 Publications Verification
Cat. No.: HY-14879B
CAS No.: 2938989-90-1
Purity:  98.66%
Synonyms: NXL-104 hydrate; AVE1330A hydrate
Research Areas:  

Infection

Avibactam sodium (NXL-104) hydrate is a covalent and reversible non-β-lactam β-lactamase inhibitor which inhibits β-lactamase TEM-1 and CTX-M-15 with IC50s of 8 nM and 5 nM, respectively [1].
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11
11 Cited Publications
Cat. No.: HY-120859
CAS No.: 1436861-97-0
Purity:  99.32%
Synonyms: WCK-5107
Zidebactam (WCK-5107) is a potent β-lactamase inhibitor . Zidebactam also is a penicillin-binding protein2 (PBP2) inhibitor with an IC50 of 0.26 μg/mL .
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9
9 Cited Publications
Cat. No.: HY-106178
CAS No.: 219639-75-5
Purity:  99.98%
Synonyms: 3D53
PMX-53 (3D53) is a synthetic peptidic and a potent and orally active complement C5a receptor (CD88) antagonist with an IC50 of 20 nM. PMX-53 is also a low-affinity MrgX2 agonist that stimulates MrgX2-mediated mast cell degranulation. PMX-53 specifically binds to C5aR1 and does not bind to the second C5aR (C5L2) and C3aR. PMX-53 has anti-inflammatory, anticancer and antiatherosclerotic effects [1] .
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3
3 Cited Publications
Cat. No.: HY-P0227
CAS No.: 168482-23-3
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

SHU 9119 is a potent human melanocortin 3 and 4 receptors (MC3/4R) antagonist and a partial MC5R agonist; with IC50 values of 0.23, 0.06, and 0.09 nM for human MC3R, MC4R and MC5R, respectively.
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2
2 Cited Publications
Cat. No.: HY-B1434
CAS No.: 957-68-6
Synonyms: 7-ACA
7-aminocephalosporanic acid (7-ACA) is a HSP90β inhibitor and an antibiotic. 7-Aminocephalosporanic acid is the core chemical structure of the synthesis of cephalosporin antibiotics and an effective β-lactamase inhibitor .
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1
1 Cited Publications
Cat. No.: HY-P0267
CAS No.: 121062-08-6
Melanotan (MT)-II is a melanocortin receptor agonist. Melanotan (MT)-II activates melanocortin receptor 3 and melanocortin receptor 4, and stimulates the release of central endogenous oxytocin. Melanotan (MT)-II reverses recognition memory impairment, increased anxiety levels and reduced exploratory tendency in zebrafish exposed to short-term high-fat diet. Melanotan (MT)-II improves impaired social behavior indicators in mouse models of autism spectrum disorder. Melanotan (MT)-II induces weight loss, reduces food intake and exerts anorectic effects. Melanotan (MT)-II increases intracavernous pressure and erectile activity in brown rats. Melanotan (MT)-II can be used in studies related to memory impairment, anxiety, reduced exploratory behavior, autism spectrum disorder, obesity and erectile dysfunction [1] .
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1
1 Cited Publications
Cat. No.: HY-18678A
CAS No.: 1607799-13-2
Synonyms: PT-141 Acetate
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

Bremelanotide (PT-141) Acetate is a melanocortin receptor agonist. Bremelanotide Acetate can activate MC4R and increases dopamine release. Bremelanotide Acetate induces appetitive sexual behaviors, female mounting behavior, and repetitive self-grooming. Bremelanotide Acetate can be used for the research of hypoactive sexual desire disorders [1] .
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1
1 Cited Publications
Cat. No.: HY-A0248A
CAS No.: 4135-11-9
Polymyxin B1 is a potent antimicrobial lipopeptide first derived from Bacilus polymyxa. Polymyxin B1 is the major component in Polymyxin B (HY-A0248). Polymyxin B1 can induce lysis of bacterial cells through interaction with their membranes. Polymyxin B1 has the potential for multidrug-resistant Gram-negative bacterial infections treatment [1] .
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Cat. No.: HY-145632
CAS No.: 2538014-94-5
Synonyms: ALT-801
Target:  

GLP Receptor GCGR

Research Areas:  

Metabolic Disease

Pemvidutide (ALT-801) is a GLP-1R/GCGR dual agonist, shows striking reductions in body weight, liver fat and serum lipids. Pemvidutide can be used in non-alcoholic steatohepatitis (NASH) and obesity research [1].
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Cat. No.: HY-14879AR
CAS No.: 1192491-61-4
Synonyms: NXL-104 (Standard)
Avibactam (sodium) (Standard) is the analytical standard of Avibactam (sodium). This product is intended for research and analytical applications. Avibactam sodium (NXL-104) is a covalent and reversible non-β-lactam β-lactamase inhibitor which inhibits β-lactamase TEM-1 and CTX-M-15 with IC50s of 8 nM and 5 nM, respectively [1].
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Cat. No.: HY-14879S2
Synonyms: NXL-104-13C5
Avibactam sodium salt- 13C5 (NXL-104- 13C5) is 13C labeled Avibactam (sodium). Avibactam sodium (NXL-104) is a covalent and reversible non-β-lactam β-lactamase inhibitor which inhibits β-lactamase TEM-1 and CTX-M-15 with IC50s of 8 nM and 5 nM, respectively [1] .
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Cat. No.: HY-P11290
CAS No.: 1228015-10-8
Target:  

Melanocortin Receptor

Research Areas:  

Metabolic Disease

MC4-NN2-0453, a α-MSH analog, is a selective MC4R agonist. MC4-NN2-0453 can be used for obesity research [1].
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Cat. No.: HY-P10447
CAS No.: 103651-09-8
Synonyms: FengycIN IX; SNA-60-367-3
Target:  

Phospholipase Fungal

Research Areas:  

Infection

Plipastatin A1 (Fengycin IX; SNA-60-367-3) is a lipopeptide with phospholipase A2 inhibitory activity. Plipastatin A1 inhibits conidial germination of Botrytis cinerea in vitro and reduces the incidence of gray mold on tomato leaves. Plipastatin A1 is applicable to research related to gray mold [1][2].
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Cat. No.: HY-136306
CAS No.: 1087784-71-1
Purity:  99.60%
Research Areas:  

Infection

Metallo-beta-lactamase ligand 1 is a class B β-lactamase inhibitor with antibacterial activity extracted from patent WO2019221122A1, compound A [1].
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Cat. No.: HY-P1208
CAS No.: 667430-81-1
Target:  

Melanocortin Receptor

Research Areas:  

Inflammation/Immunology

PG-931, an analog of SHU 9119 (HY-P0227), is a potent melanocortin 4 (MC4) receptor (IC50=0.58 nM) agonist and is more selective than for the hMC3R (IC50=55 nM) or the hMC5R (IC50=2.4 nM). PG-931 can reverse haemorrhagic shock and prevent multiple organ damage in vivo .
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Cat. No.: HY-A0248AS
Polymyxin B1-d7 TFA is the deuterium labeled Polymyxin B1 TFA (HY-A0248A). Polymyxin B1 is a potent antimicrobial lipopeptide first derived from Bacilus polymyxa. Polymyxin B1 is the major component in Polymyxin B (HY-A0248). Polymyxin B1 can induce lysis of bacterial cells through interaction with their membranes. Polymyxin B1 has the potential for multidrug-resistant Gram-negative bacterial infections treatment [1] .
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Cat. No.: HY-145632A
Purity:  98.07%
Synonyms: ALT-801 TFA
Target:  

GLP Receptor GCGR

Research Areas:  

Metabolic Disease

Pemvidutide (ALT-801) TFA is a GLP-1R/GCGR dual agonist, shows striking reductions in body weight, liver fat and serum lipids. Pemvidutide TFA can be used in non-alcoholic steatohepatitis (NASH) and obesity research [1].
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