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Results for "

carbazole derivatives

" in MedChemExpress (MCE) Product Catalog:
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Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-108637
    PhiKan 083
    1 Publications Verification

    		 MDM-2/p53 Cancer
    PhiKan 083 is a carbazole derivative, which binds to the surface cavity and stabilizes Y220C (a p53 mutant), with a Kd of 167 μM. PhiKan 083 can be used for cancer research .
    PhiKan 083
  • HY-135776
    BMVC2

    o-BMVC

    		 G-quadruplex Cancer
    BMVC2 (o-BMVC) is a bisubstitute carbazole derivative of BMVC. BMVC2 is a G-quadruplex (G4) stabilizer .
    BMVC2
  • HY-108510
    Rimcazole dihydrochloride

    BW 234U dihydrochloride

    		 Sigma Receptor Dopamine Receptor Neurological Disease Cancer
    Rimcazole (BW 234U) dihydrochloride is a carbazole derivative that acts in part as a sigma (σ) receptor antagonist. Rimcazole dihydrochloride also binds with moderate affinity to the dopamine transporter and inhibit dopamine uptake. Rimcazole dihydrochloride can reduce locomotor activity and sensitization. Rimcazole dihydrochloride also can be used for the research of cancer .
    Rimcazole dihydrochloride
  • HY-W022224
    3,6-Diiodo-9H-carbazole
    1 Publications Verification

    		 Endogenous Metabolite Others
    3,6-Diiodo-9H-carbazole is an organic compound that can be used for the design and synthesis of carbazole derivatives .
    3,6-Diiodo-9H-carbazole
  • HY-148179
    Neuropeptide Y5 receptor ligand-1

    		Neuropeptide Y Receptor Neurological Disease
    Neuropeptide Y5 receptor ligand-1 (compound 54), a carbazole derivative, is a potent neuropeptide Y5 (NPY-5) receptor antagonist .
    Neuropeptide Y5 receptor ligand-1
  • HY-108637A
    PhiKan 083 hydrochloride
    1 Publications Verification

    		 MDM-2/p53 Cancer
    PhiKan 083 hydrochloride is a carbazole derivative, which binds to the surface cavity and stabilizes Y220C (a p53 mutant), with a Kd of 167 μM , and a relative binding affinity (Kd) of 150 μM in Ln229 cells .
    PhiKan 083 hydrochloride
  • HY-U00323
    Carbazole derivative 1

    2-Fluoro-7-[(3-pyridinyl)methyl]-9H-carbazole

    		 Drug Derivative Androgen Receptor Estrogen Receptor/ERR Endocrinology
    Carbazole derivative 1 is a carbazole derivative which can be used to reduce androgen or oestrogen levels in mammals, including humans.
    Carbazole derivative 1
  • HY-163775
    Anti-inflammatory agent 88

    		MyD88 NF-κB Inflammation/Immunology
    Anti-inflammatory agent 88 (compound 6) is a carbazole derivative with anti-inflammatory activity found in marine Streptomyces. It exerts its anti-inflammatory effect by inhibiting pro-inflammatory factors and enhancing the expression of anti-inflammatory factors in the Myd88/Nf-κB pathway. Anti-inflammatory agent 88 can be used for the development of anti-inflammatory drugs .
    Anti-inflammatory agent 88
  • HY-108637R
    PhiKan 083 (Standard)

    		Reference Standards MDM-2/p53 Cancer
    PhiKan 083 (Standard) is the analytical standard of PhiKan 083 (HY-108637). This product is intended for research and analytical applications. PhiKan 083 is a carbazole derivative, which binds to the surface cavity and stabilizes Y220C (a p53 mutant), with a Kd of 167 μM. PhiKan 083 can be used for cancer research .
    PhiKan 083 (Standard)
  • HY-108510R
    Rimcazole dihydrochloride (Standard)

    BW 234U dihydrochloride (Standard)

    		 Reference Standards Sigma Receptor Dopamine Receptor Neurological Disease Cancer
    Rimcazole dihydrochloride (Standard) is the analytical standard of Rimcazole (dihydrochloride) (HY-108510). This product is intended for research and analytical applications. Rimcazole (BW 234U) dihydrochloride is a carbazole derivative that acts in part as a sigma (σ) receptor antagonist. Rimcazole dihydrochloride also binds with moderate affinity to the dopamine transporter and inhibit dopamine uptake. Rimcazole dihydrochloride can reduce locomotor activity and sensitization. Rimcazole dihydrochloride also can be used for the research of cancer .
    Rimcazole dihydrochloride (Standard)
  • HY-179523
    Carba1

    		Drug Derivative NAMPT Microtubule/Tubulin Neurological Disease Cancer
    Carba1 is a bifunctional Carbazole (HY-D0204) derivative that activates nicotinamide phosphoribosyltransferase (NAMPT) and enhances NAD biosynthesis. Carba1 binds to colchicine site of tubulin, enhancing the anti-tumor effect of various chemotherapy drugs, such as Paclitaxel (HY-B0015). Carba1 exerts neuroprotective effect and can regulate cell energy metabolism. Carba1 can be used for the researches of cancer and chemotherapy-induced peripheral neuropathy (CIPN) .
    Carba1
  • HY-179670
    Antibacterial agent 304

    		Bacterial Infection
    Antibacterial agent 304 (Compound 3a) is an antibacterial agent with a minimum inhibitory concentration (MIC) of 8 μg/mL against S. aureus and P. aeruginosa. This antibacterial agent has a bactericidal effect and can disrupt the integrity of the cell wall. Antibacterial agent 304 has the potential to be a sustainable organic photocatalyst .
    Antibacterial agent 304

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