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Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!2025-02-06
16 Results for "
peripheral benzodiazepine receptor
" in MedChemExpress (MCE) Product Catalog:
Products (16)
16 Results for "peripheral benzodiazepine receptor" in MCE Product Catalog:
1
1 Cited Publications
Cat. No.: HY-19945
CAS No.: 220551-92-8
Target:
Research Areas:
DAA1106 is a peripheral benzodiazepine receptor (PBR) agonist that is permeable to the blood-brain barrier, but has no affinity for GABAA receptors.
Cat. No.: HY-W013150
CAS No.: 82626-01-5
Target:
Research Areas:
Alpidem, an anxiolytic agent, is an orally active and brain-penetrant GABAA receptor ligand, binds to α1β2γ2 subunit-containing GABAA receptors (IC50 of 17 nM) over α5β2γ2 subunit-containing GABAA receptors (IC50 of >10 μM). Alpidem modulates calcium-induced mitochondrial permeability transition, induces glutathione depletion and hepatocyte necrosis, potentiates TNF-α toxicity, inhibits marble-burying and locomotor activity, enhances stressed rodent feeding behavior, and exerts anticonvulsant effects. Alpidem can be used for the research of anxiety, anxiety disorders, and convulsions .
Target:
Research Areas:
FGIN 1-27, an indoleacetamide, is a specific peripheral benzodiazepine receptor (PBR) ligand with a Ki of 5.0 nM. FGIN 1-27 can penetrate the blood brain barrier (BBB). FGIN 1-27 inhibits the onset of Isoniazid-induced convulsions .
Cat. No.: HY-A0198
CAS No.: 37115-32-5
Synonyms: U 41123
Target:
Research Areas:
Adinazolam (U 41123) is a triazolobenzodiazepine. Adinazolam binds to peripheral-type benzodiazepine receptors which interact allosterically with GABA receptors. Adinazolam has dual anxiolytic and antidepressant activities .
Cat. No.: HY-119605
CAS No.: 220551-79-1
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DAA-1097 is an orally active and selective agonist for the peripheral benzodiazepine receptor (PBR). DAA-1097 has anxiolytic effects .
Cat. No.: HY-118096
CAS No.: 109960-13-6
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Research Areas:
AHN 070 is an irreversible peripheral benzodiazepine receptor (PBR) ligand. AHN 070 can bind to PBR with nanomolar affinity and is pH-dependent. AHN 070 can be used for studying the structure and function of PBR .
Cat. No.: HY-101059R
CAS No.: 142720-24-9
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Research Areas:
FGIN 1-27 (Standard) is the analytical standard of FGIN 1-27. This product is intended for research and analytical applications. FGIN 1-27, an indoleacetamide, is a specific peripheral benzodiazepine receptor (PBR) ligand with a Ki of 5.0 nM. FGIN 1-27 can penetrate the blood brain barrier (BBB). FGIN 1-27 inhibits the onset of Isoniazid-induced convulsions .
Cat. No.: HY-118308
CAS No.: 143934-15-0
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AHN-683 is a luciferin-derived ligand that targets the peripheral benzodiazepine receptor (BDR).
Cat. No.: HY-A0198A
CAS No.: 57938-82-6
Synonyms: U 41123F mesylate
Target:
Research Areas:
Adinazolam (U 41123F) mesylate is a triazolobenzodiazepine. Adinazolam mesylate binds to peripheral-type benzodiazepine receptors which interact allosterically with GABA receptors. Adinazolam mesylate has dual anxiolytic and antidepressant activities .
Cat. No.: HY-A0198S
Synonyms: U 41123-d5
Cat. No.: HY-P702478
Purity: ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: Tspo; Bzrp; Mbr; Translocator protein; Mitochondrial benzodiazepine receptor; PKBS; peripheral-type benzodiazepine receptor; PBR; PBS; PBRS; PTBR; BPBS; Translocator Protein (18kDa); Benzodiazapine receptor (peripheral); benzodiazepine peripheral Binding
Species:
Mouse
Source:
E. coli Cell-free
Cat. No.: HY-P87004
Synonyms: Benzodiazapine receptor (peripheral) antibody; benzodiazepine peripheral binding site antibody; BPBS antibody; BZRP antibody; DBI antibody; IBP antibody; Isoquinoline carboxamide-binding protein antibody; MBR antibody; mDRC antibody; Mitochondrial benzodiazepine receptor antibody; Benzodiazapine receptor (peripheral) antibody; benzodiazepine peripheral binding site antibody; BPBS antibody; BZRP antibody; DBI antibody; IBP antibody; Isoquinoline carboxamide-binding protein antibody; MBR antibody; mDRC antibody; Mitochondrial benzodiazepine receptor antibody; PBR antibody; PBS antibody; peripheral benzodiazepine receptor antibody; peripheral benzodiazepine receptor-related protein antibody; peripheral type benzodiazepine receptor antibody; peripheral-type benzodiazepine receptor antibody; pk18 antibody; PKBS antibody; PTBR antibody; Ptbzr antibody; PTBZR02 antibody; RATPTBZR02 antibody; translocator protein (18kDa) antibody; Translocator protein antibody; Tspo antibody; Tspo1 antibody; TSPOA_HUMAN antibody;
Cat. No.: HY-P706194
Purity: ≥ 90%, as determined by reducing SDS-PAGE.
Synonyms: Translocator protein; Mitochondrial benzodiazepine receptor; PKBS; peripheral-type benzodiazepine receptor; PBR
Species:
Human
Source:
E. coli Cell-free
Cat. No.: HY-W436366
CAS No.: 220448-02-2
Research Areas:
SSR180575 is a specific and potent peripheral benzodiazepine receptor ligand. SSR180575 irreversibly and specifically binds with high affinity on rat heart mitochondria (Kd = 1.95 nM). SSR180575 can be used in the research of cardiovascular diseases .
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Protocols
Targeted therapy! The Capetin Prize winning "Click Chemistry" can be used like this!Targeted therapy! The Nobel Prize winning "Click Chemistry" can be used like this!A suitable model is crucial in drug screening experiments. Organs can mimic the three-dimensional functional structure of internal organs, have similar spatial organization to corresponding organs, maintain some key characteristics, and reproduce some physiological functions. They are widely used for modeling and personalized drug screening physiological functions.2025-02-06
