1. Membrane Transporter/Ion Channel
    Neuronal Signaling
    GPCR/G Protein
  2. Calcium Channel
    5-HT Receptor
  3. Nexopamil racemate

Nexopamil racemate 

Cat. No.: HY-101727
Handling Instructions

Nexopamil racemate is the racemate of Nexopamil. Nexopamil is a combined Ca2+/5-HT2 antagonist on thrombus formation in vivo and on platelet aggregation in vitro.

For research use only. We do not sell to patients.

Nexopamil racemate Chemical Structure

Nexopamil racemate Chemical Structure

CAS No. : 116759-35-4

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Description

Nexopamil racemate is the racemate of Nexopamil. Nexopamil is a combined Ca2+/5-HT2 antagonist on thrombus formation in vivo and on platelet aggregation in vitro.

IC50 & Target

5-HT2 Receptor

 

Ca2+

 

In Vitro

Serotonin-induced platelet aggregation in dog platelet-rich plasma (PRP) in vitro is most potently inhibited by Nexopamil (IC50 81 nM) [1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

In Vivo

Nexopamil (0.05 mg/kg) completely abolishes cyclic flow reductions (CFRs) during the first 30 min after application without significantly altering hemodynamics[1].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Molecular Weight

404.59

Formula

C₂₄H₄₀N₂O₃

CAS No.
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Storage

Please store the product under the recommended conditions in the Certificate of Analysis.

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Product Name:
Nexopamil racemate
Cat. No.:
HY-101727
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