2. シグナル伝達
  3. GPCR/G Protein
  4. Kisspeptin Receptor
  5. Kisspeptin Receptor Antagonist

Kisspeptin Receptor Antagonist

Kisspeptin Receptor Antagonists (4):

製品番号 製品名 製品効果 純度
  • HY-P1196A
    Kisspeptin 234 TFA Antagonist 98.92%
    Kisspeptin 234 TFA, is a 10 amino acid peptide as well as a kisspeptin receptor (KISS1, GPR54) antagonist. Kisspeptin 234 TFA is an analog of Kisspeptin 10.
  • HY-182421
    GPR54 antagonist-1 Antagonist
    GPR54 antagonist‑1 is a GPR54 antagonist with IC50 values of 3.6 nM and 15 nM against human and rat GPR54, respectively. GPR54 antagonist‑1 shows blood‑brain barrier penetration. GPR54 antagonist‑1 blocks the function of human and rat GPR54 receptors. GPR54 antagonist‑1 suppresses plasma luteinizing hormone levels in castrated male rats. GPR54 antagonist‑1 can be used for the study of prostate cancer and endometriosis.
  • HY-P11341
    Kisspeptin antagonist p271 Antagonist 99.76%
    Kisspeptin antagonist p271 is a Kisspeptin antagonist with cell-penetrating ability. Kisspeptin antagonist p271 can block the binding of endogenous Kisspeptin to GPR54 on pituitary somatotropes, thereby relieving the inhibition of growth hormone secretion. Kisspeptin antagonist p271 can specifically and significantly stimulate growth hormone secretion, while inhibiting luteinizing hormone without affecting prolactin or cortisol. Kisspeptin antagonist p271 can be used in the research of diseases related to insufficient growth hormone secretion.
  • HY-P1196
    Kisspeptin 234 Antagonist
    Kisspeptin 234, is a 10 amino acid peptide as well as a kisspeptin receptor (KISS1, GPR54) antagonist. Kisspeptin 234 is an analog of Kisspeptin 10.