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Cat. No.: HY-136878

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LSD1-IN-10

LSD1-IN-10 is a LSD1/MAO inhibitor with LSD1 IC₅₀ of 5 nM, MAO-A IC₅₀ of 16 μM, and MAO-B IC₅₀ of 7.4 μM. LSD1-IN-10 suppresses enzymatic activity of LSD1, MAO-A, and MAO-B. LSD1-IN-10 can be used for the research of cancer, alzheimer's disease, parkinson's disease, huntington's disease.

Nos produits utilisent uniquement pour la recherche. Nous ne vendons pas aux patients.

CAS No.: 1235864-15-9
Formule: C₁₉H₂₁NO₂
Masse moléculaire:295.38

Stockage:

Please store the product under the recommended conditions in the Certificate of Analysis.

LSD1-IN-10 Chemical Structure

CAS No.: 1235864-15-9

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Fluorescent Dye

Strong Fluorescence Signal / Multi-Disciplinary Applications / High Fluorescence Specificity

Activité biologique
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références
Calculators
Help & FAQs
Classifications
Bioz

Activité biologique

Description

IC₅₀ & Target^[1]

LSD1

5 nM (IC₅₀)

MAO-A

16 μM (IC₅₀)

MAO-B

7.4 μM (IC₅₀)

Voir tous les produits spécifiques à Isoform Histone Demethylase :

Voir tous les produits spécifiques à Isoform Monoamine Oxidase :

MAO-A
MAO-B

In Vitro

LSD1-IN-10 (Compound 76) potently inhibits LSD1 with an IC₅₀ of 0.005 μM, and is far less potent against MAO-A (IC₅₀ 16 μM) and MAO-B (IC₅₀ 7.4 μM) in cell-free enzymatic assays^[1].

MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only.

Chemical Information

CAS No. 1235864-15-9
Masse moléculaire 295.38
Formule C₁₉H₂₁NO₂
SMILES

N(C(C)C=1C=C2C(=CC1)OCCO2)[C@H]3[C@@H](C3)C4=CC=CC=C4
Livraison

Room temperature in continental US; may vary elsewhere.
Stockage

Please store the product under the recommended conditions in the Certificate of Analysis.

Pureté et documentation

Instruction de manipulation (2659 KB)

Références

[1]. Nathalie G, et al. Phenylcyclopropylamine derivatives and their medical use. United States, WO2010084160 A. 2010-07-29.

Calculators

Calculateur de molarité

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

Mass Mass

Concentration Concentration

Volume Volume

Molecular Weight Molecular Weight

Calculateur de dilution

Concentration _(start) × Volume _(start) = Concentration _(final) × Volume _(final)

Concentration _(start) Concentration _(start)

Volume _(start) Volume _(start)

Concentration _(final) Concentration _(final)

Volume _(final) Volume _(final)

Help & FAQs

How should lyophilized recombinant proteins be reconstituted and stored?

1. Before opening the cap, centrifuge the vial at 13000 rpm for 20-30 seconds. This step will ensure that any lyophilized powder that may have adhered to the cap or walls is collected at the bottom of the vial, minimizing the risk of product loss.

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MOQ

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100 mg

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Activité biologique
- Description
- IC₅₀ & Target
- In Vitro
Chemical Information
Pureté et documentation
Références

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LSD1-IN-10

Voir tous les produits spécifiques à Isoform Histone Demethylase

Voir tous les produits spécifiques à Isoform Monoamine Oxidase

Activité biologique

Chemical Information

Pureté et documentation

Références

Calculators

Help & FAQs

LSD1-IN-10 Related Classifications

HY-136878 Related Classifications