120493-42-7
Chemical Structure
GEA 857
- CAS No.: 120493-42-7
- Formula:C15H22ClNO2
- Molecular Weight:283.79
IUPAC Name: 1-(4-chlorophenyl)-2-methylpropan-2-yl L-valinate
InChIKey: YKRSWMGPYKJOBF-ZDUSSCGKSA-N
SMILES: N[C@@H](C(C)C)C(OC(C)(C)CC1=CC=C(Cl)C=C1)=O
Biological Activity: GEA 857 is a structural analog of the Serotonin (HY-B1473A) uptake blocker Alaproclate (HY-164011). GEA 857 enhances responses induced by muscarinic receptor agonists by inhibiting certain calcium-dependent potassium channels on membranes, a blockade that can enhance or prolong the muscarinic cholinergic effects. GEA 857 can be used in research on neurodegenerative diseases[1].
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GEA 857 | GEA 857 is a structural analog of the Serotonin (HY-B1473A) uptake blocker Alaproclate (HY-164011). GEA 857 enhances responses induced by muscarinic receptor agonists by inhibiting certain calcium-dependent potassium channels on membranes, a blockade that can enhance or prolong the muscarinic cholinergic effects. GEA 857 can be used in research on neurodegenerative diseases. | |||||||||||||||||||||
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Keywords
