2400958-08-7
Chemical Structure
BJP-06-005-3
- CAS No.: 2400958-08-7
- Formula:C37H48ClN7O7
- Molecular Weight:738.27
IUPAC Name: ethyl (S)-2-((S)-2-((S)-1-(N-(2-chloroacetyl)-N-methyl-L-phenylalanyl)piperidine-2-carboxamido)-3-(1H-indol-3-yl)propanamido)-5-ureidopentanoate
InChIKey: SUAZSPTYLUTEDZ-ORYMTKCHSA-N
SMILES: O=C([C@H]1N(CCCC1)C([C@@H](N(C)C(CCl)=O)CC2=CC=CC=C2)=O)N[C@H](C(N[C@H](C(OCC)=O)CCCNC(N)=O)=O)CC3=CNC4=CC=CC=C34
Biological Activity: BJP-06-005-3 is a selective Pin1 inhibitor with a Ki value of 48 nM. BJP-06-005-3 induces the degradation of mutant KRAS. BJP-06-005-3 inhibits pancreatic ductal adenocarcinoma via the Pin1-mediated pathway. BJP-06-005-3 is used in studies related to KRAS-mutant pancreatic ductal adenocarcinoma[1][2].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
BJP-06-005-3 | BJP-06-005-3 is a selective Pin1 inhibitor with a Ki value of 48 nM. BJP-06-005-3 induces the degradation of mutant KRAS. BJP-06-005-3 inhibits pancreatic ductal adenocarcinoma via the Pin1-mediated pathway. BJP-06-005-3 is used in studies related to KRAS-mutant pancreatic ductal adenocarcinoma. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
