MDL-102234
MDL-102234 is a potent and selective adenosine A1 receptor antagonist with a Ki value of 23.2 nM at the adenosine A1 receptor. MDL-102234 can be used for the study of cognition enhancement-related neural functions.
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- CAS No.: 137766-81-5
- Formule: C20H26N4O2
- Masse moléculaire:354.45
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
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Activité biologique
Description
IC50 & Target
[1]|
A1AR 23.2 nM (Ki) |
In Vitro
MDL-102234 (tested in receptor binding assays) (26 °C) exhibits high binding affinity to adenosine A1 receptor (Ki = 23.2 nM) and low binding affinity to adenosine A2 receptor (Ki = 3510 nM), with an A2/A1 selectivity ratio of 153[1].
MedChemExpress (MCE) has not independently confirmed the accuracy of these methods. They are for reference only. .
Chemical Information
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CAS No. 137766-81-5
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Masse moléculaire 354.45
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Formule C20H26N4O2
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SMILES
CCCN1C2=C(C(N(C1=O)CCC)=O)NC([C@@H](C3=CC=CC=C3)CC)=N2
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
MDL-102234 Related Classifications
HY-182518 Related Classifications
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