TASP0412098
TASP0412098 is an orally available, potent and selective CRTH2/DP2 antagonist with high binding affinity (IC50 2.1 nM) and functional activity (IC50 12 nM). TASP0412098 has the potential to suppress asthma in mouse and guinea pig bronchial asthma models.
For research use only. We do not sell to patients.
- CAS No.: 1233248-29-7
- Formula: C27H23ClN2O3
- Molecular Weight:458.94
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
CRTH2/DP2[1]
Chemical Information
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CAS No. 1233248-29-7
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Molecular Weight 458.94
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Formula C27H23ClN2O3
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SMILES
O=C(CC1=CN=C(C2=C1C=CC=C2)CC3=CC=C(C=C3)C(NCCC4=CC=C(C=C4)Cl)=O)O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)