ER covalent antagonist-1
ER covalent antagonist-1 (Compound 39D) is the antagonist for estrogen receptor α (ERα). ER covalent antagonist-1 inhibits the proliferation of ERα-positive cell MCF-7 with an IC50 of 0.98 μM, arrests the cell cycle at G0/G1 phase, and induces apoptosis. ER covalent antagonist-1 exhibits antitumor efficacy in mouse model.
For research use only. We do not sell to patients.
- CAS No.: 2757498-74-9
- Formula: C33H32N2O5S
- Molecular Weight:568.68
-
Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
-
Biological Activity
-
Chemical Information
- Purity & Documentation
- References
-
Help & FAQs
Biological Activity
Chemical Information
-
CAS No. 2757498-74-9
-
Molecular Weight 568.68
-
Formula C33H32N2O5S
-
SMILES
O=C(C1=CC=CC=C1)C(SC2=CC(O)=CC=C23)=C3OC4=CC=C(C=C4)OC5CN(C5)C/C=C/C(N6CCCCC6)=O
-
Shipping
Room temperature in continental US; may vary elsewhere.
-
Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
ER covalent antagonist-1 Related Classifications
HY-170382 Related Classifications
Powered by Bioz